Lus Taw Qhia
99 feem pua dasatinib hmoov yog ib yam ntawm qhov ncauj muaj me me-molecule multikinase inhibitor. Tsis tsuas yog nws zoo txwv BCR-ABL thiab SRC-tsev neeg kinases (SRC, LCK, YOG, FYN), tab sis kuj inhibit C-KIT, PDGFR- thiab , thiab ephrin receptor kinase. Cov tshuaj no tau raug pov thawj tias nws muaj zog tiv thaiv kev hloov pauv hauv kev kho mob, suav nrog kev kho Imatinib. Cov mis mos molecular ntawm cov khoom yog C22H26ClN7O2S, qhov hnyav molecular yog 488.006, thiab solubility yog 35.35 mg / mL. Nws feem ntau yog grey rau daj khoom.
Cov txiaj ntsig
99 feem pua dasatinib hmoov yog ib hom inhibitor ntawm ntau yam tyrosine kinase, suav nrog BCR-ABL kinase ntsig txog mob granulocytic leukemia thiab lwm yam mob qog noj ntshav. Nws tsuas yog kho mob ntev, ceev myeloid lossis lymphoblastic mob myeloid leukemia hauv cov laus. Tsis tas li ntawd, nws tuaj yeem kho cov tsos mob uas tiv taus imatinib. Cov khoom no yog siv los kho cov neeg laus uas muaj Philadelphia chromosome positive (Ph plus) chronic myeloid leukemia (CML) uas tiv taus imatinib mesylate lossis cov uas tsis kam ua rau nws nyob rau hauv lub sijhawm ntev, nrawm thiab mob hnyav (mob myeloid thiab mob lymphocytic)

Cov duab ntxaws

Specification
PSA | 134.75000 | LogP | 2.24 |
EINECS | 801-607-0 | CAS | 302962-49-8 |
Cov khoom pom zoo
99% Dasatinib Hmoov | Efitinib | TIAB SA 195 |
Ibrutinib | TIAB SA 9291 | Lapatinib |
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FAQ
1. Qhov kev pom zoo npaum li cas?
Rau cov neeg mob uas muaj CML mob ntev: 100-140mg ib hnub, ib hnub ib zaug, noj qhov ncauj.
Rau cov neeg mob uas muaj lymphocytic leukemia siab heev los yog Ph chromosome zoo (PhXxX) mob lymphocytic leukemia: 70-100mg ib hnub, ib hnub ib zaug, noj qhov ncauj.
Txog cov koob tshuaj kom raug, ua raws li koj tus kws kho mob cov lus qhia.
2. Puas muaj kev sib tham nrog tshuaj?
Txhawm rau kom cov tshuaj muaj txiaj ntsig zoo, tsis txhob siv cov tshuaj hauv qab no: CYP3A4 inhibitor, anti acid, thiab proton twj tso kua mis inhibitor.
Yog tias koj txaus siab rau peb cov khoom, thov koj xav tiv tauj peb ncaj qha.
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