Kev mob yog lub teeb liab ntshiab - qhov hnyav, feem ntau crippling ceeb toom los ntawm lub cev. Thaum mob mob heev tshwm sim, txawm tias los ntawm kev raug mob, kev phais mob, lossis mob o, tau txais kev pab sai thiab muaj txiaj ntsig zoo. DExKetoprofofofofen yog qhov kev xaiv kho mob loj uas muab kev pabcuam tam sim ntawd thiab txiav txim siab. Raws li cov ntshiab nquag enantiomer ntawm ketoprofen, nws zam kev hloov pauv metabolic thiab tuaj yeem ua tiav cov nyhuv analgesic. Hauv kev sib tham no, peb yuav tshawb xyuas cov tshuab ntawm kev ua, chaw kuaj mob cov kev pab cuam, thiab siv daim ntawv thov kho ntawm DEXKETOPROPENFE.
Dab tsi yog dexketoprofen
Dexketoprofren 99 hmoovYog cov lus tsis txaus ntseeg -} kub (nsaid) feem ntau siv los kho luv- mob hnyav thiab mob. Nws paub rau nws txoj kev ua kom zoo thiab ua tau zoo vim yog Ketoprofen ("txoj cai} Qhov no txhais tau tias koj lub cev tsis tas yuav hloov nws kom pib muab kev mob siab. Kev mob siab yog tam sim ntawd, khaus, thiab luv {{6} nyob. Nws pab daws qhov o, liab, thiab ua npaws tshwm sim los ntawm kev mob hauv lub cev. Piv nrog lwm NSAIDs, nws kuj tuaj yeem txo ua npaws. Yog tias koj txaus siab rau dexkessoprofofofofrofen, thov tsis txhob ua siab deb hu rau Xi'an Sonwu rau peb txoj kev ua hauj lwm ncaj qha.

Li cas dexoneploppen ua haujlwm
Dexkessoprofen inhibits cyclooxygarease (COx) enzymes, tshwj xeeb Cox-1 thiab Cox-2, yog li txo cov prostaglandins. Prostaglandins yog thawj qhov ua rau kub taub hau, o, thiab malaise. Nws cov kev nquag ua haujlwm enantiomer ua tau zoo rau kev mob qis dua thiab muaj qhov nrawm dua ntawm kev ua haujlwm ntau dua li kev sib cais ketoprofen. Nws cov tshuab ntawm kev ua yog raws li hauv qab no:
1. COx enzyme inhibition
DExKymoprofofrofen inhibits cov kev ua si ntawm cyclooxyenase enzymes (tshwj xeeb yog Cox-1 thiab Cox-2). Cov enzymes no yuav tsum muaj rau kev tsim cov prostaglandins, uas yog tsim los ntawm lub cell membrane tivthaiv Archar.
2. Txo cov khoom lag luam prostaglandin ntau lawm
Cox inhibitors durastically txwv Prostaglandin ntau lawm. Prostaglandins muaj cov tshuaj hormone - zoo li lwg me uas pab ntau yam ua haujlwm hauv lub cev. Lawv sensitize txoj hlab ntaws rau kev mob siab, ua rau cov hlab ntshav (dilation ntawm cov hlab ntshav), nce ntshav ntws, thiab ua rau o thiab liab. Lawv tseem ua raws li hypothalamus (lub hlwb cov kev tswj kub (lub hlwb cov kev tswj kub), stimulating mucus thiab bicarbonate ntau lawm (COX-1 hais txog).
3. Kho cov teebmeem
Nws ua haujlwm los ntawm kev txo cov rhiab rau qhov mob -}}}}}}}}}}} itectagins uas ua rau o thiab liab. Los ntawm kev txo cov prostaglandins hauv hypothalamus, nws yog qhov tshwj xeeb rau kev mob me, xws li mob kaus hniav, mob tus leeg, thiab mob nqaij tus mob.
4. "Dex -" dominance (enantiomer tshwj xeeb)
Nws yog cov nquag enantiomer (txoj cai - lias molecule) ntawm cov kab kev sib xyaw ntawm Ketoprofen. Tsuas yog daim foos tshwj xeeb no tsuas yog ua tau zoo nyob rau hauv inhibiting COX enzymes. Kev xa tawm tsuas yog nquag enantiomer tso cai rau qhov quav qis kom ua tiav cov nyhuv tib yam, nrog kev ua kom sai dua ntawm kev nqis tes ua. Qhov no muaj kev txo qis rau kis rau cov tsis muaj zog enantiomer, yog li txo cov tshuaj uas yuav ua rau cov kev mob tshwm sim.

Yog dexketoprofofofofen tib yam li ibuprofen
Tsis yog, dexkessoprofof deg tsis zoo ib yam li ibuprofen. Thaum lawv koom nrog tib chav kawm cov tshuaj thiab qhia qee qhov zoo sib xws, lawv muaj ob yam tshuaj sib txawv nrog qhov sib txawv. Cov khoom no yog muaj zog dua, nrawm dua {} Ua yeeb tshuaj uas yuav tsum tau siv rau kev mob nkeeg (NSAIL) Ibuprofen, ntawm qhov tod tes, yog ib qho zoo - paub, generic, tshaj {} conter {} stere reducer. Nws yog thawj qhov kev xaiv rau kev hloov kho txhua hnub thiab mob.
Hauv qab no yog cov ncauj lus piav qhia ntxiv ntawm lawv.

1. Chemically, cov khoom no tsis yog ib qho tseem ceeb ntawm ibuprofen tab sis tus dextrorotatory enantiomer ntawm Ketoprofen. Nws yog cov qauv sib txawv ntawm cov qauv qub uas cuam tshuam rau nws cov khoom siv tshuaj pharmacological.
2. Nyob rau hauv cov nqe lus ntawm potency thiab kev siv, dexkessoprofofofofofofofof 25 mg koob tshuaj tuaj yeem ua tiav kev ua tau zoo piv rau, lossis ntau dua kev ua tau zoo dua, cov tshuaj ntau dua ntawm ibuprofen (piv txwv li, 200-400 mg).
3. Tsis tas li ntawd, Dexketoprofofofen ua yeeb yam tshiab siv thiab pib ua haujlwm, feem ntau ua rau mob hnyav kom tau kev mob sai. Ibuprofen, ntawm qhov tod tes, muaj qhov qeeb zuj zus ntawm kev nqis tes ua.
4. Nyob rau hauv cov nqe lus ntawm muaj, ob qho txawv cuam tshuam: ibuprofen muaj nyob rau hauv ob qho qis {2} {{{{{{{} {dose tshuaj; Txawm li cas los xij, vim nws cov khoom muaj ntau dua thiab cov khoom lag luam, cov khoom lag luam no yog cov tshuaj hauv feem ntau thiab xav tau kws kho mob cov lus qhia.
5. Txawm hais tias ob qho tib si muaj cov kev mob nsaid zoo sib xws, lawv txawv hauv zaus thiab siv.
Dab tsi yog qhov zoo ntawm dexketoprofofrofen
Nws yog lub vas nrawm- ua yeeb tshuaj nrog kev sib xyaw ua ke, ua rau nws tsim nyog rau kev kuaj mob kom ua pa nrawm. Nws tseem ceeb analgesic cov phiaj xwm zoo heev relieves ntau yam mob thiab lwm yam mob me me mus rau mob nqaij tawv,
Kev mob hniav, thiab dysmenorrhea, ntawm lwm cov ua rau mob. Nws qhov tseem ceeb luv luv ntawm kev ua (feem ntau yog plaub mus rau teev) tso cai rau kev siv hluav taws xob, tso cai rau kev hloov kho rau txhua tus neeg mob xav tau.
Raws li cov kws tshuaj ua haujlwm nquag s (+) enantiomer ntawm ketoprofen, nws ua rau muaj kev sib tw ntau dua li cov kev sib zog ntawm cov tshuaj qis, uas pab txhim kho kev tsim nyog thiab kev nyab xeeb.
Txog rau cov lus nug txog DEXKETOPROFOFOFOFOFORCEN 99 hmoov tus nqi, lossis lwm yam khoom {{{}}}}}}} sonwu ncaj qha.
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