Dab tsi yog Compounded Itraconazole
R51211 hmoovyog ib hom tshuaj uas tsim tshwj xeeb rau kev siv hauv tsiaj los kho cov kab mob fungal. Nws yog nyob rau hauv chav kawm ntawm triazole antifungal agents thiab feem ntau yog muab los ntawm kws kho tsiaj los kho ntau yam kab mob fungal nyob rau hauv dev, miv, thiab lwm yam tsiaj.
Itraconazole hmoov yog tsim tshwj xeeb rau cov kws kho tsiaj siv thiab tuaj yeem ua cov hmoov nplej uas tuaj yeem sib xyaw ua ke hauv ntau hom, xws li kev ncua lossis tshuaj pleev, nyob ntawm tus neeg mob xav tau. Qhov kev hloov pauv no tso cai rau kev noj tshuaj thiab kev tswj hwm raws li cov cai tshwj xeeb ntawm txhua tus tsiaj.
Cov tshuaj ua haujlwm los ntawm inhibiting cov synthesis ntawm ergosterol, ib qho tseem ceeb ntawm cov kab mob fungal cell membranes, zoo tiv thaiv kev loj hlob thiab kis ntawm fungus. Nws muaj ntau yam kev ua ub no tiv thaiv ntau hom fungi, nrog rau cov kab mob dermatophytes, cov poov xab, thiab cov pwm feem ntau pom nyob rau hauv cov kab mob veterinary fungal.
Veterinary itraconazole hmoov feem ntau yog siv los kho cov kab mob fungal, xws li blastomycosis, histoplasmosis, thiab cryptococcosis. Nws tseem muaj txiaj ntsig zoo hauv kev tswj cov kab mob fungal zoo li kab mob hauv cov tsiaj.
Kev noj tshuaj kom raug thiab kev tswj hwm ntawm itraconazole hmoov yog qhov tseem ceeb rau kev pom zoo. Qhov ntau npaum li cas yog txiav txim los ntawm tus kws kho tsiaj raws li hom thiab qhov hnyav ntawm tus kab mob fungal, nrog rau tus tsiaj tus yam ntxwv. Nws yog ib qho tseem ceeb uas yuav tsum tau ua raws li kws kho tsiaj cov lus qhia kom meej kom paub meej tias cov tshuaj raug muab.

Certificate of Analysis
|
SAIB |
SPECIFICATION |
TSEEM CEEB |
|
Qhov tshwm sim |
Dawb los yog yuav luag dawb hmoov |
Yuav luag dawb hmoov |
|
Kev txheeb xyuas |
IR ua raws li tus qauv |
Ua raws |
|
Qhov tshwm sim ntawm kev daws teeb meem |
Kev daws S yog qhov tseeb thiab tsis muaj xim ntau dua li siv tshuaj R6 lossis B6 |
Ua raws |
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Cov khoom muaj feem xyuam |
|
|
|
Cov impurities B |
Tsis ntau tshaj 0.3 feem pua |
Tsis pom |
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Cov impurities G |
Tsis ntau tshaj 0.3 feem pua |
0.1 feem pua |
|
Impurity E |
Tsis ntau tshaj 0.2 feem pua |
Tsis pom |
|
Qhov sib npaug ntawm impurities C thiab D |
Tsis ntau tshaj 0.3 feem pua |
Tsis pom |
|
Unspecified impurities |
Tsis ntau tshaj 0.10 feem pua |
0.06 feem pua |
|
Tag nrho impurities |
Tsis ntau tshaj 0.8 feem pua |
0.3 feem pua |
|
Poob rau ziab |
Tsis ntau tshaj 0.5 feem pua |
0.1 feem pua |
|
Sulfated tshauv |
Tsis ntau tshaj 0.10 feem pua |
0.03 feem pua |
|
Assay |
99.0 feem pua rau 101.0 feem pua |
99.12% ua |
Qhov twg Yuav Itraconazole Powder
Xi'an Sonwu muaj kev paub dhau los hauv kev lag luam thoob ntiaj teb thiab kev noj qab haus huv kev lag luam. Credit-raws li thiab zoo ua ntej yog lub hauv paus ntsiab lus ntawm Xi'an Sonwu tuam txhab. Xi'an Sonwu nruj me ntsis tswj cov khoom zoo, yog li kev xaiv pib nrog cov khoom siv raw. Tsis tas li ntawd, peb tswj txhua qhov kev nthuav dav thiab txo cov nqi kom peb cov neeg siv khoom tuaj yeem tau txais cov khoom lag luam zoo tshaj plaws. Raws li cov no, cov neeg siv khoom tau txais kev qhuas siab rau peb cov khoom. Yog li nrhiav Xi'an Sonwu Biotech Co., Ltd.
Xi'an Sonwu tag nrho ua kom cov khoom zoo, yog li cov qauv tuaj yeem muab tau. Ntawm no yog qhov ntau.
|
Daim ntawv |
Tus Qauv Zauv |
Yam tsawg kawg nkaus |
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Hmoov |
500g |
1kg ua |
Cov neeg siv khoom 'Cov lus pom zoo

Dab tsi yog Itraconazole Siv Hauv Tsiaj
Itraconazole yog siv dav siv tshuaj tua kab mob hauv cov kws kho tsiaj. Nws belongs rau chav kawm triazole ntawm cov tshuaj thiab muaj txiaj ntsig zoo tiv thaiv ntau yam kab mob fungal hauv cov tsiaj. Ntawm no yog saib ze dua ntawm kev siv itraconazole hauv ntau hom.
1. Cov dev:
- Aspergillosis: Itraconazole feem ntau yog siv los kho cov kab mob ua pa thiab aspergillosis hauv cov dev, uas tshwm sim los ntawm cov kab mob Aspergillus. Qhov no tuaj yeem yog qhov nyuaj rau kev kho mob, thiab itraconazole feem ntau suav hais tias yog tshuaj ntawm kev xaiv.
- Blastomycosis: Itraconazole yog ib feem tseem ceeb ntawm kev kho mob rau blastomycosis, kab mob fungal tshwm sim los ntawm Blastomyces dermatitidis.
- Histoplasmosis: Cov kab mob fungal no tshwm sim los ntawm Histoplasma capsulatum tuaj yeem cuam tshuam rau dev, thiab itraconazole feem ntau yog siv los ua thawj kab.
- Dermatophytosis: Itraconazole zoo tiv thaiv qee hom dermatophytes, uas ua rau cov kab mob ringworm hauv dev. Nws feem ntau yog siv raws li kev kho mob thib ob thaum lwm cov tshuaj tsis zoo lossis tsis zoo.
- Cryptococcosis: Itraconazole tuaj yeem siv los tswj cov kab mob cryptococcal hauv cov dev, tshwj xeeb tshaj yog nyob rau hauv cov xwm txheej uas fluconazole tsis zoo lossis zam.
2. miv:
- Cryptococcosis: Itraconazole yog ib qho kev kho mob tseem ceeb rau cov kab mob cryptococcal hauv miv, tshwj xeeb tshaj yog rau cov kab mob hauv lub cev.
- Dermatophytosis: Zoo ib yam li dev, itraconazole tuaj yeem siv los kho cov kab mob ringworm hauv miv.
- Aspergillosis: Hauv miv, itraconazole tuaj yeem siv los tswj qhov ntswg lossis nthuav tawm aspergillosis.
3. Nees:
- Kab mob fungal: Itraconazole tuaj yeem siv los kho ntau yam kab mob fungal hauv cov nees, suav nrog aspergillosis thiab coccidioidomycosis.
4. Noog:
- Aspergillosis: Avian hom, tshwj xeeb tshaj yog cov noog ntawm prey, tuaj yeem raug rau aspergillosis. Itraconazole feem ntau siv los kho cov kab mob fungal no hauv cov noog.

Ntev npaum li cas rau Itraconazole ua haujlwm hauv dev
Lub sijhawm nws siv rauR51211 hmoovmus ua hauj lwm hauv dev tuaj yeem sib txawv nyob ntawm ntau yam, nrog rau hom thiab qhov hnyav ntawm cov kab mob fungal raug kho. Nws yog ib qho tseem ceeb kom nkag siab tias kev kho tshuaj tiv thaiv kab mob feem ntau yuav tsum tau siv sijhawm ntev kom ua tiav qhov kev daws teeb meem ntawm tus kab mob thiab nws cov tsos mob tshwm sim. Nov yog qee cov ntsiab lus tseem ceeb hais txog lub sijhawm rau itraconazole los siv rau cov dev:
1. Lub sij hawm rau cov lus teb thawj zaug: Qee zaum, cov dev yuav pom kev txhim kho nyob rau thawj ob peb hnub mus rau lub lis piam ntawm kev pib kho itraconazole. Qhov no tuaj yeem tshwm sim raws li kev txo qis hauv cov tsos mob xws li cov kab mob ntawm daim tawv nqaij, cov tsos mob ua pa, lossis lwm yam tshwm sim ntawm tus kab mob fungal. Txawm li cas los xij, nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias kev txhim kho pom tsis tas yuav qhia txog kev tshem tawm tag nrho ntawm tus kab mob.
2. Lub sij hawm kho mob: Cov kab mob fungal hauv cov dev feem ntau yuav tsum tau ncua sij hawm kho mob txij li lub lis piam mus rau hli. Lub sijhawm ntawm kev kho mob nrog itraconazole nyob ntawm ntau yam, nrog rau hom fungus koom nrog, qhov chaw thiab thaj tsam ntawm tus kab mob, thiab tus neeg teb cov lus teb ntawm tus dev. Koj tus kws kho tsiaj yuav txiav txim siab lub sijhawm kho kom haum raws li cov kev xav no.
3. Cov kab mob fungal: Rau cov kab mob fungal, xws li blastomycosis, histoplasmosis, lossis aspergillosis, kev kho mob nrog itraconazole feem ntau kav ntev li ob peb lub hlis. Cov kab mob no tuaj yeem nyuaj rau kev kho mob, thiab nws tseem ceeb heev uas yuav tsum tau siv tshuaj ntxiv raws li koj tus kws kho tsiaj tau sau tseg, txawm tias koj tus dev cov tsos mob zoo dua. Kev txiav tawm ntxov ntxov ntawm kev kho mob tuaj yeem ua rau rov qab los yog tsis tiav kev daws teeb meem ntawm tus kab mob.
4. Ringworm (dermatophytosis): Ringworm yog kab mob fungal uas cuam tshuam rau ntawm daim tawv nqaij, plaub hau, lossis rau tes. Kev kho mob nrog itraconazole rau ringworm feem ntau kav ntev li ob peb lub lis piam mus rau ob peb lub hlis. Kev saib xyuas tsis tu ncua ntawm daim tawv nqaij thiab plaub hau rau kev txhim kho kev kho mob, nrog rau kev rov ua cov kab mob fungal, yog qhov tseem ceeb los xyuas kom meej tias tus kab mob tau daws tag nrho.
5. Kev mus ntsib kws kho mob: Thaum kho nrog itraconazole, nws yog ib qho tseem ceeb uas yuav tau ua raws li kev mus ntsib kws kho mob tsis tu ncua. Cov kev mus ntsib no tso cai rau kev soj ntsuam zoo ntawm tus dev qhov kev nce qib, saib xyuas cov kev mob tshwm sim lossis kev hloov pauv hauv cov ntshav, thiab hloov kho cov kev kho mob yog tias xav tau.
6. Teb variability: Nws yog ib qho tseem ceeb kom nkag siab tias tus dev ib leeg thiab cov kab mob fungal sib txawv tuaj yeem teb txawv rau kev kho mob itraconazole. Yog li ntawd, lub sij hawm teb yuav txawv. Qee tus dev yuav xav tau kev kho mob ntev dua ua ntej pom kev txhim kho tseem ceeb, thaum lwm tus tuaj yeem teb sai dua. Kev ua siab ntev thiab ua raws li koj tus kws kho tsiaj cov lus qhia yog qhov tseem ceeb ntawm txoj haujlwm no.
Nco ntsoov tias kev kho mob ua tiav tsis yog tsuas yog tshem tawm tus kab mob xwb tab sis kuj tswj hwm cov xwm txheej hauv qab no, xws li kev tiv thaiv kev tiv thaiv kab mob lossis ib puag ncig, txhawm rau tiv thaiv kev rov ua dua lossis rov ua dua tshiab.
Yog Itraconazole Zoo dua Ketoconazole Rau Cov dev
Thaum muab piv rau itraconazole thiab ketoconazole rau kev kho cov kab mob fungal hauv dev, ntau yam yuav tsum tau xav txog. Ob qho tshuaj yog cov tshuaj tua kab mob thiab koom nrog tib chav kawm ntawm cov tshuaj, azole antifungals. Txawm li cas los xij, muaj qee qhov sib txawv ntawm lawv uas tuaj yeem cuam tshuam lawv cov txiaj ntsig thiab kev tsim nyog rau kev siv dev.
1. Spectrum ntawm kev ua ub no: Itraconazole feem ntau muaj ib tug dav spectrum ntawm antifungal kev ua si piv rau ketoconazole. Nws muaj txiaj ntsig zoo tiv thaiv ntau yam kab mob, suav nrog Aspergillus, Blastomyces, Histoplasma, thiab Cryptococcus. Ketoconazole, ntawm qhov tod tes, feem ntau zoo tiv thaiv kab mob dermatophytes (ringworm) thiab Malassezia hom, tab sis nws yuav tsis zoo li kev tiv thaiv kab mob los yog kab mob fungal.
2. Kev ua tau zoo: Hais txog kev ua tau zoo, itraconazole feem ntau suav tias muaj txiaj ntsig zoo dua li ketoconazole rau qee yam kab mob fungal hauv dev. Piv txwv li, aspergillosis, blastomycosis, thiab histoplasmosis feem ntau yog tswj tau zoo dua nrog itraconazole vim nws lub zog ntau dua thiab kev ua haujlwm dav dav.
3. Kev nyab xeeb profile: Ob qho tib si itraconazole thiab ketoconazole tuaj yeem muaj cov kev mob tshwm sim, tab sis itraconazole nyiam ua kom zoo dua los ntawm cov dev. Ketoconazole muaj feem cuam tshuam nrog kev pheej hmoo siab dua ntawm kev tsis zoo, suav nrog kev mob plab hnyuv, mob siab rau lub siab, txo qis qab los noj mov, thiab kev sib cuam tshuam ntawm cov tshuaj. Itraconazole, thaum feem ntau muaj kev nyab xeeb, tseem tuaj yeem ua rau mob plab hnyuv thiab qee zaus cuam tshuam rau daim siab ua haujlwm. Kev saib xyuas tsis tu ncua yog ib qho tseem ceeb thaum siv ob qho tshuaj.
Pharmacokinetics: Itraconazole muaj qhov ncauj bioavailability zoo dua piv rau ketoconazole, txhais tau tias nws nqus tau zoo dua thiab ua tiav qib siab hauv cov hlab ntsha. Qhov no tso cai rau kom zoo dua faib rau cov ntaub so ntswg thiab txhim kho kev kho mob.

Dab tsi yog Cov Teeb Meem Ntawm Itraconazole Hauv Cov dev
Itraconazole feem ntau tau txais txiaj ntsig zoo hauv cov dev, tab sis zoo li txhua yam tshuaj, nws tuaj yeem muaj qee yam kev phiv. Nws yog ib qho tseem ceeb kom paub txog cov kev mob tshwm sim no thiab saib xyuas koj tus dev kom zoo thaum kho. Nov yog qee qhov ua tau tshwm sim ntawm itraconazole hauv dev:
1. Kev cuam tshuam ntawm plab hnyuv: Qhov feem ntau tshwm sim ntawm itraconazole nyob rau hauv dev muaj feem xyuam rau txoj hnyuv. Cov no yuav muaj xws li txo qis qab los noj mov, ntuav, raws plab, lossis cov quav mos. Cov tsos mob no feem ntau yog mob me me thiab ntuav, thiab feem ntau lawv tuaj yeem tswj tau los ntawm kev tswj hwm cov tshuaj nrog noj mov lossis txo qhov ntau npaum li cas.
2. Hepatotoxicity: Itraconazole muaj peev xwm ua rau lub siab puas tsuaj rau qee tus dev. Lub siab enzymes (piv txwv li, alanine aminotransferase, alkaline phosphatase) tuaj yeem pom ntawm cov ntshav. Kev saib xyuas lub siab ua haujlwm los ntawm kev kuaj ntshav tsis tu ncua yog qhov tseem ceeb thaum kho. Yog hais tias lub siab enzyme nce siab tshwm sim, kev txiav tawm ntawm itraconazole yuav tsum yog qhov tsim nyog.
3. Hypoadrenocorticism (Addison tus kab mob): Muaj tsawg zaus, itraconazole tau txuam nrog kev loj hlob ntawm hypoadrenocorticism hauv dev. Qhov xwm txheej no ua rau txo qis cov tshuaj hormones steroid los ntawm cov qog adrenal. Cov tsos mob tuaj yeem suav nrog kev qaug zog, qaug zog, tsis qab los noj mov, ntuav, poob phaus, lossis kab mob plab. Yog tias cov tsos mob no tshwm sim, nws yog ib qho tseem ceeb kom nrhiav kev kho mob sai sai.
4. Cov tsos mob ntawm lub paj hlwb: Txawm tias tsis tshua muaj tshwm sim, itraconazole tau txuas rau cov tsos mob ntawm cov hlab ntsha hauv qee tus dev. Cov no tuaj yeem suav nrog ataxia (tsis muaj kev sib koom tes), tshee, qaug dab peg, lossis lwm yam kev coj cwj pwm txawv txav. Yog tias pom muaj cov tsos mob neurological, nws tseem ceeb heev kom tiv tauj koj tus kws kho tsiaj tam sim ntawd.
5. Kev tsis haum tshuaj: Muaj tsawg zaus, dev yuav muaj kev fab tshuaj rau itraconazole. Cov tsos mob ntawm kev tsis haum tshuaj tej zaum yuav muaj xws li lub ntsej muag o, khaus, khaus, ua tsis taus pa, los yog vau. Yog tias koj tus dev pom cov tsos mob ntawm kev tsis haum tshuaj, nrhiav kev kho tsiaj tam sim ntawd.
6. Kev sib cuam tshuam tshuaj: Itraconazole tuaj yeem cuam tshuam nrog qee yam tshuaj, suav nrog qee cov tshuaj tiv thaiv kab mob, tshuaj tiv thaiv kab mob, lossis lwm yam tshuaj tua kab mob. Nws yog ib qho tseem ceeb kom qhia rau koj tus kws kho tsiaj txog txhua yam tshuaj uas koj tus dev noj kom tsis txhob muaj kev cuam tshuam tshuaj.
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