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API Hmoov Cilostazol

API Hmoov Cilostazol

Cov tsos mob: Dawb Crystals Hmoov
Specification: 99%
CAS: 73963-72-1
Cov roj formula: C20H27N5O2
Molecular Luj: 369.46
Txee Lub neej: 2 Xyoo Kev Cia Siab
Tshuag: Tsim nyog Tshuag
Daim ntawv pov thawj: COA, ISO, GMP, HACCP, SGS
Kev Pabcuam: Kev Pabcuam OEM (Pub Private Package)

Khoom Taw qhia

 

Yam tshuaj twg yog Cilostazol
API hmoov cilostazoleyog ib qho tshuaj antiplatelet feem ntau yog siv los kho qhov sib cuam tshuam claudication los ntawm atherosclerosis. Nws tiv thaiv phosphodiesterase III (PDE3) los ntawm kev ua haujlwm, uas nce intracellular cyclic adenosine monophosphate (cAMP) qib thiab ua rau vasodilation thiab platelet aggregation kom nres. Hauv luv luv, nws pab txhim kho cov ntshav khiav thiab txo qhov mob ceg thiab tsis xis nyob, tshwj xeeb tshaj yog thaum taug kev. Nws tuaj yeem kho cov tsos mob ischemic tshwm sim los ntawm cov kab mob atherosclerosis ntev, nthuav cov hlab ntsha, txhim kho cov hlab ntsha peripheral, thiab txo cov tsos mob xws li mob, mob, ua daus no, thiab claudication. Nws tiv thaiv kev rov tshwm sim ntawm cerebral infarction, muaj cov nyhuv antiplatelet aggregation, thiab tuaj yeem hloov cov tshuaj xws li aspirin lossis clopidogrel.
Cov tshuaj no feem ntau yog siv los txhim kho cov teeb meem ntshav ncig los ntawm kab mob peripheral arterial tab sis kuj tuaj yeem kho lwm yam kab mob plawv. Vim nws ob qho kev cuam tshuam ntawm vasodilation thiab antiplatelet, nws tuaj yeem pab cov neeg mob nce kev taug kev deb thiab txo qis cov tsos mob tshwm sim los ntawm cov ntshav tsis zoo. Yog li, Xi'an Sonwu tuaj yeem muab cov ntaub ntawv nyoos cilostazol.

Cilostazol structure

 

Certificate Of Analysis

Cov khoom tsom xam

Specification

Cov qhabnias xeem

Kev ntsuam xyuas (HPLC)

98.0%-102.0%

99.39%

Qhov tshwm sim

Dawb mus rau dawb crystals hmoov

Dawb crystals hmoov

Solubility

Dawb soluble hauv chloroform; me ntsis soluble hauv methanol thiab cawv; xyaum insoluble hauv dej.

Ua tau raws li qhov yuav tsum tau ua

Kev txheeb xyuas

A: Infrared spectrum yuav tsum ua raws li IR spectrum ntawm cilostazol ua haujlwm tus qauv.

Ua raws

B: Lub sijhawm khaws cia ntawm lub ncov loj hauv chromatogram ntawm kev tshuaj ntsuam kev npaj sib raug rau qhov hauv chromatogram ntawm tus qauv npaj, raws li tau txais hauv qhov kev xeem.

Ua raws

Poob rau ziab

Tsawg dua lossis sib npaug rau 0.3%

0.13%

Residue ntawm ignition

Tsawg dua lossis sib npaug rau 0.1%

0.04%

Chlorides

Tsawg dua los yog sib npaug rau 0.018%

Ua raws

Yam khoom

A: Tsawg dua lossis sib npaug rau 0.1%

B: Tsawg dua lossis sib npaug rau 0.1%

C: Tsawg dua lossis sib npaug rau 0.1%

Ib qho impurity Tsawg dua lossis sib npaug rau 0.1%

Tag nrho cov imurities Tsawg dua lossis sib npaug rau 0.4%

Ua raws

Ua raws

Ua raws

Ua raws

Ua raws

Tag nrho cov phaj suav

NMT 1, 000cfu/ml

Ua raws

Poov & pwm

NMT 100cfu/ml

Ua raws

Sakmonella

Tsis zoo

Tsis zoo

E.coli

Tsis zoo

Tsis zoo

Tag nrho cov phaj suav

NMT 1, 000cfu/ml

Ua raws

 

Yuav Cilostazol
Xi'an Sonwu Biotech Co. Ltd. muaj ntau tshaj kaum xyoo ntawm kev lag luam kev lag luam, tshwj xeeb hauv kev tsim thiab muag cov ntaub ntawv raw. Xi'an Sonwu tau tsim kev sib koom tes ruaj khov thiab txhim khu kev qha nrog cov teb chaws hauv Asmeskas, Asia, Europe, thiab Oceania. Xi'an Sonwu muab cov khoom zoo ua ntej thiab siv zog los muab txhua tus neeg siv khoom nrog cov kev pabcuam zoo kom tau raws li lawv cov kev xav tau tag nrho.
Cov khoom lag luam zoo yog Xi'an Sonwu qhov tseem ceeb tshaj plaws, thiab lub tuam txhab kev mob siab rau kev ua tiav tau pom nyob rau hauv txhua yam ntawm nws cov haujlwm, suav nrog kev xaiv cov khoom siv raw, cov txheej txheem tsim khoom, cov qauv kuaj, thiab cov neeg ua haujlwm tshaj lij. Los ntawm kev tswj hwm txhua qhov kev nthuav dav, Xi'an Sonwu tuaj yeem txo tus nqi yam tsis muaj kev cuam tshuam zoo, ua kom cov neeg siv khoom tau txais cov khoom muaj txiaj ntsig tshwj xeeb.
Xi'an Sonwu zoo siab rau cov lus pom zoo uas nws tau txais los ntawm cov neeg siv khoom, uas tau lees paub qhov zoo ntawm cov khoom. Txhawm rau ua pov thawj ntxiv cov khoom lag luam, Xi'an Sonwu yuav muab cov qauv rau koj los kuaj.

Daim ntawv

Tus Qauv Zauv

MOQ

Hmoov

100g

100g


Cov neeg siv khoom 'Cov lus pom zoo

-1001

 

Yog Cilostazol Ib Ntshav Thinner lossis Anticoagulant
Nws tsis yog ib txwm ntshav thinner lossis anticoagulant. Nws raug cais raws li tus neeg sawv cev antiplatelet. Cov tshuaj antiplatelet tiv thaiv platelets los ntawm clumping ua ke, ib qho ntawm thawj kauj ruam hauv kev tsim cov ntshav txhaws. Hauv qhov sib piv, cov tshuaj tiv thaiv coagulants zoo li warfarin lossis heparin cuam tshuam nrog cov hlab ntsha los tiv thaiv cov ntshav txhaws los ntawm kev tsim. Nws lub luag haujlwm tseem ceeb ntawm kev ua haujlwm cuam tshuam nrog inhibiting ib qho enzyme hu ua phosphodiesterase III (PDE3), uas ua rau nce cyclic AMP (cAMP) qib hauv platelets thiab vascular du leeg.
Inhibition of Platelet Aggregation: Nws txo qhov kev pheej hmoo ntawm cov hlab ntsha los ntawm kev tiv thaiv platelets los ntawm kev ua ke.
Vasodilation: Nws so thiab nthuav cov hlab ntsha, tshwj xeeb tshaj yog nyob rau hauv ob txhais ceg, txhim kho cov ntshav khiav.
Yog li ntawd, thaum nws pab tiv thaiv cov ntshav txhaws, nws yog qhov txawv ntawm cov tshuaj tiv thaiv coagulants thiab tau muab faib ua cov tshuaj antiplatelet.

 

Dab tsi yog Cov Txheej Txheem Ntawm Kev Ua Ntawm Cilostazol
Cov txheej txheem ntawm kev ua ntawm nws feem ntau cuam tshuam nrog inhibition ntawm phosphodiesterase III (PDE3). PDE3 yog ib qho tseem ceeb enzyme nyob rau hauv tsev neeg phosphodiesterase (PDE) thiab tseem ceeb heev rau kev tswj cov txheej txheem intracellular signaling. PDE3 feem ntau rhuav tshem ob lub cim tseem ceeb ntawm lub cev: cyclic adenosine monophosphate thiab cyclic guanosine monophosphate. Hais txog nws cov teebmeem ntawm platelets, PDE3 tswj cov qib cAMP hauv platelets, cuam tshuam rau platelet aggregation. PDE3 inhibitors siv cov tshuaj tiv thaiv kab mob los ntawm kev nce qib cAMP thiab inhibiting platelet activation thiab aggregation. Qhov no inhibition ua rau ob lub ntsiab pharmacological cuam tshuam: inhibition ntawm platelet aggregation thiab vasodilation.
Nws inhibits PDE3, thiab los ntawm inhibiting PDE3, nws nce intracellular cAMP qib. Nce cAMP txo platelet aggregation (coagulation) thiab txhawb kev so ntawm vascular du nqaij. Nce cAMP hauv platelets txo lawv lub peev xwm los lo ua ke, txo qhov kev pheej hmoo ntawm thrombus tsim. Qhov no yog tshwj xeeb tshaj yog pab tau rau kev tiv thaiv arterial thrombosis. Kev nce cAMP kuj ua rau kom cov leeg nqaij du, tshwj xeeb tshaj yog nyob rau hauv cov hlab ntsha peripheral. Qhov no vasodilation txhim kho cov ntshav khiav, tshwj xeeb tshaj yog rau ob txhais ceg, ua rau nws muaj txiaj ntsig zoo rau kev sib cuam tshuam claudication (mob los ntawm cov ntshav tsis txaus mus rau qhov kawg).

Mechanism Of Action Of Cilostazol

 

Kev siv Cilostazol
1. Antiplatelet nyhuv
API hmoov cilostazolence cyclic adenosine monophosphate (cAMP) qib hauv platelets thiab txo platelet adhesion thiab aggregation los ntawm inhibiting phosphodiesterase III (PDE3). Qhov ntawd pab tiv thaiv cov ntshav txhaws thiab tshwj xeeb tshaj yog pab kho thiab tiv thaiv kab mob arteriosclerotic.

Antiplatelet effect

2. Cov nyhuv vasodilation
Kev nce qib cAMP hauv cov leeg nqaij du ua rau vasodilation, uas ua rau cov leeg nqaij du. Cov nyhuv no tseem ceeb tshwj xeeb hauv cov hlab ntsha peripheral, xws li cov hlab ntsha hauv ob txhais ceg, txhim kho cov ntshav khiav thiab yog li txo cov tsos mob tshwm sim los ntawm cov kab mob peripheral arterial, xws li tsis sib haum xeeb claudication (kev mob ceg thaum taug kev).

3. Txhim kho kev muaj peev xwm kis las
Nws ua haujlwm los ntawm kev nthuav dav cov hlab ntsha peripheral thiab tiv thaiv platelet aggregation, txhim kho lub neej zoo thiab tsis mob taug kev deb rau cov neeg uas muaj kev sib cuam tshuam claudication.

4. Anti-atherosclerotic nyhuv
Nws muaj peev xwm tiv thaiv platelet aggregation thiab nthuav cov hlab ntsha, txo cov kev pheej hmoo ntawm cov hlab plawv thiab cerebrovascular txheej xwm thiab kev loj hlob thiab tsim ntawm atherosclerotic plaques.

5. Txhim kho lub plawv ua haujlwm
Txawm hais tias nws tsuas yog siv rau cov kab mob peripheral arterial, nws yuav muaj txiaj ntsig zoo inotropic ntawm lub plawv ua haujlwm (txhim kho myocardial contractility) los ntawm kev nce qib myocardial cell cAMP, uas yuav pab tau qee cov neeg mob plawv tsis txaus. Pab tau.

6. Anti-inflammatory thiab anti-proliferative teebmeem

enhancing myocardial contractility

Nws kuj tau pom tias muaj cov tshuaj tiv thaiv tshwj xeeb thiab inhibitory cuam tshuam rau vascular du leeg cell proliferation, uas tej zaum yuav muaj txiaj ntsig zoo hauv kev tiv thaiv thiab kho arteriosclerosis thiab nws cov teeb meem.

 

Dab tsi yog Qhov Kev Tsis Pom Zoo rau Cilostazol
Nws tuaj yeem ua rau qee qhov kev mob tshwm sim thaum siv tshuaj kho mob. Txawm hais tias feem ntau cov neeg mob tuaj yeem zam tau lawv, qee qhov kev mob tshwm sim yuav xav tau kev saib xyuas tshwj xeeb lossis kev cuam tshuam.
Cov teebmeem tshwm sim
Kev mob taub hau yog ib qho ntawm cov kev mob tshwm sim feem ntau, uas feem ntau cuam tshuam nrog vasodilation nyhuv ntawm cov tshuaj.
Nws tuaj yeem ua rau mob plab tsis zoo, thiab qee zaum, nws yog ib qho tsim nyog yuav tsum tau kho cov zaub mov lossis tshuaj noj.
kiv taub hau kuj tshwm sim, uas tej zaum yuav cuam tshuam rau vasodilation thiab ntshav siab-txo cov teebmeem.
Vim tias cov tshuaj tuaj yeem ua rau lub plawv dhia nce ntxiv, qee cov neeg mob yuav hnov ​​​​lub plawv dhia nrawm lossis palpitations.
Qee cov neeg mob tej zaum yuav muaj ceg lossis pob qij txha edema, uas feem ntau cuam tshuam nrog vasodilation nyhuv ntawm cov tshuaj.

 

Cov teebmeem loj
Vim tias nws tuaj yeem ua rau lub plawv dhia nce ntxiv, cov teeb meem no yuav ua rau cov neeg mob mob plawv mob hnyav (xws li lub plawv tsis ua haujlwm lossis mob arrhythmia). Cov neeg mob uas muaj lub plawv tsis ua hauj lwm hnyav yuav tsum tsis txhob noj nws vim tias nws tuaj yeem ua rau muaj kev pheej hmoo ntawm cov hlab plawv.
Vim nws cov nyhuv antiplatelet, nws yuav ua rau muaj kev pheej hmoo los ntshav, tshwj xeeb tshaj yog thaum siv nrog lwm cov tshuaj antiplatelet (xws li tshuaj aspirin thiab clopidogrel) los yog anticoagulants (xws li warfarin). Qhov chaw los ntshav ntau: los ntshav cov pos hniav, qhov ntswg, tawv nqaij, thiab lwm yam.

 

Lwm yam kev mob tshwm sim tsis tshua muaj tshwm sim
Qhov muag tsis pom kev tuaj yeem cuam tshuam nrog vasodilation lossis cuam tshuam rau lub paj hlwb.
Txo qab los noj mov yuav ua rau me ntsis poob phaus.
Vim yog vasodilation, qee cov neeg mob yuav muaj mob me ntsis hypotension.

Adverse Reaction To Cilostazol

 

Hoobkas
1. Xi'an Sonwu Biotech Co., Ltd muaj nws lub Hoobkas los tsim, tsim, thiab khaws cov khoom, yog li muaj cov khoom tsim nyog. Xi'an Sonwu muaj kev txiav txim kom zoo, huv si, thiab huv si ntau lawm. Nyob rau hauv Xi'an Sonwu, cov kws tshawb fawb tuaj yeem tsim cov khoom tshiab zoo.
2. Xi'an Sonwu muaj cov cai nruj rau cov neeg ua haujlwm faib los ntawm kev tsim khoom thiab kev sim rau kev muag khoom. Txhawm rau kom ntseeg tau tias txhua yam khoom raug thauj mus los, kev txhawb nqa cov ntaub ntawv nruj thiab kev pabcuam tom qab muag tau muab.

factory


Daim ntawv pov thawj

certificates

 

Ntim

packaging

 

Logistics

-1002

Dhau li lav cov khoom, lwm qhov tseem ceeb tshaj plaws yog cov neeg siv khoom tuaj yeem tau txais cov khoom zoo. Yog li, Xi'an Sonwu muab txhua yam kev xa khoom raws li kev xav tau sib txawv.

courier

 

FAQ
1. Lub zog muaj zog
Xi'an Sonwu Owning muaj lub chaw tsim khoom, OEM Hoobkas, thiab chav kuaj.
2. Muaj kev paub
Ua lag luam xa tawm thoob plaws ntiaj teb rau ntau tshaj kaum xyoo.
3. Pab neeg tshaj lij
Xi'an Sonwu muaj pab pawg muag khoom thiab kev pabcuam zoo.
4. Kev Pabcuam Siab Siab
Xi'an Sonwu muaj pab pawg muag khoom thiab kev pabcuam zoo. Xi'an Sonwu Tau nyob hauv kev lag luam tau ntau xyoo, cov neeg siv khoom qhuas tau mus txog 99%.
5. Cov neeg siv khoom tshuaj xyuas
Xi'an Sonwu tau nyob hauv kev lag luam tau ntau xyoo, thiab cov neeg siv khoom qhuas tau mus txog 99%.

Yog tias koj xav paub tus nqi cilostazol hmoov, koj tuaj yeem tiv tauj Xi'an Sonwu. Nyem rau email, thiab tom qab ntawd koj tau txais cov khoom zooAPI hmoov cilostazole.
Email:sales@sonwu.com

Cim npe nrov: api hmoov cilostazol, Tuam Tshoj, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, nqe, tej, ntshiab, raw, mov, kev muag khoom

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