Yam tshuaj twg yog Apremilast
Apremilast hmoovyog phosphodiesterase 4 (PDE4) inhibitor class tshuaj. Nws feem ntau kho qee yam kab mob autoimmune, suav nrog mob hnyav rau psoriasis thiab mob caj dab psoriatic. Psoriasis yog ib qho mob ntev ntawm daim tawv nqaij uas tuaj yeem rov zoo dua thiab raug coj los ntawm ntau yam, suav nrog kev tiv thaiv kab mob tsis zoo, kab mob endocrine, kab mob, thiab kab mob. Nws tsuas yog tshwm sim raws li erythema, ua daus no, mob pob qij txha, o, desquamation, thiab lwm yam. Tsis muaj kev kho mob tshwj xeeb rau psoriasis, thiab nws tuaj yeem tswj tau thiab txo qis los ntawm kev kho tshuaj, kho lub cev, thiab lwm yam. Nws relieves o, mob pob qij txha, txhav, thiab lwm yam mob tshwm sim los ntawm tus kab mob. Psoriatic mob caj dab yog ib yam kab mob uas cuam tshuam rau qee tus neeg uas muaj psoriasis thiab ua rau mob pob qij txha thiab mob. Ob qho xwm txheej tuaj yeem cuam tshuam rau lub neej zoo ntawm cov neeg cuam tshuam thiab feem ntau xav tau kev tswj xyuas mus sij hawm ntev.
Cov neeg laus uas muaj mob psoriatic mob caj dab thiab mob hnyav-rau-mob plaque psoriasis tuaj yeem coj nws. Nws ua haujlwm los ntawm kev tswj hwm cov haujlwm ntawm PDE4, ib qho enzyme uas tswj kev mob thiab kev tiv thaiv kab mob hauv lub cev. Nws cov txheej txheem ntawm kev ua haujlwm pab txo qis cov tsos mob cuam tshuam nrog cov kab mob ntev, txo cov neeg mob uas tsis tau teb lossis tsis kam rau lwm txoj kev kho mob. Yog tias koj txaus siab rau qhov inhibitor no, thov hu rau Xi'an Sonwu. Xi'an Sonwu tuaj yeem muab rau koj nrog 99- hmoov apremilast.

Certificate Of Analysis
|
Cov khoom kuaj |
Kev soj ntsuam Specification |
Cov qhabnias xeem |
|
Qhov tshwm sim |
Dawb hmoov |
Ua raws |
|
Cov khoom muaj feem xyuam |
Ib qho uas tsis paub impurity Tsawg dua lossis sib npaug rau 0.1% Tag nrho impurity Tsawg dua lossis sib npaug rau 0.5% |
0.09% 0.13% |
|
Enantiomer |
0.05% nax |
0.12% |
|
Poob rau ziab |
0.05% max |
0.03% |
|
Melting point |
154~158ºC |
Ua raws |
|
Residue ntawm ignition |
0.5% max |
0.01% |
|
Residual kuab tshuaj |
Methan ≥3000ppm Ethanol ≥5000ppm THF 720 ppm Acetonitrile ≥410ppm Aceton ≥5000ppm Dichloromethae ≥600ppm |
5 60ppm N.D. N.D. 66ppm ua 800ppm ua N.D. |
|
Assay |
99.0%min |
99.87% |
Apremilast Yuav Online
Xi'an Sonwu Biotech Co. Ltd. muaj ntau tshaj kaum xyoo ntawm kev lag luam kev lag luam, tshwj xeeb hauv kev tsim thiab muag cov ntaub ntawv raw. Xi'an Sonwu tau tsim kev sib koom tes ruaj khov thiab txhim khu kev qha nrog cov teb chaws hauv Asmeskas, Asia, Europe, thiab Oceania. Ua ntej cov khoom lag luam zoo, Xi'an Sonwu ua haujlwm nyuaj los ua kom tau raws li txhua tus neeg siv khoom xav tau los ntawm kev muab cov kev pabcuam zoo tshaj plaws.
Cov khoom lag luam zoo yog Xi'an Sonwu qhov tseem ceeb tshaj plaws, thiab lub tuam txhab kev mob siab rau kev ua tiav tau pom nyob rau hauv txhua yam ntawm nws cov haujlwm, suav nrog kev xaiv cov khoom siv raw, cov txheej txheem tsim khoom, cov qauv kuaj, thiab cov neeg ua haujlwm tshaj lij. Xi'an Sonwu tuaj yeem txo cov nuj nqis yam tsis muaj kev txi zoo los ntawm kev ua tib zoo saib xyuas txhua yam, lav tias cov neeg tau txais cov khoom muaj txiaj ntsig zoo kawg li.
Xi'an Sonwu zoo siab rau cov lus pom zoo uas nws tau txais los ntawm cov neeg siv khoom, uas tau lees paub qhov zoo ntawm cov khoom. Txhawm rau ua pov thawj ntxiv cov khoom lag luam, Xi'an Sonwu yuav muab cov qauv rau koj los kuaj.
|
Daim ntawv |
Tus Qauv Zauv |
Yam tsawg kawg nkaus |
|
Hmoov |
10g |
50g |
Cov neeg siv khoom zoo lus

Apremilast Vs Methotrexate
1. Mechanism of Action:
Apremilast: Nws yog phosphodiesterase 4 (PDE4) inhibitor. Nws ua haujlwm los ntawm inhibiting enzyme PDE4, uas koom nrog hauv cov txheej txheem inflammatory. Los ntawm kev txo qhov mob, nws pab txo cov tsos mob hauv cov mob xws li mob caj dab psoriatic thiab cov quav hniav psoriasis.
Methotrexate: Nws yog ib qho tshuaj tiv thaiv kab mob thiab tiv thaiv kab mob. Methotrexate ua haujlwm los ntawm inhibiting ib qho enzyme koom nrog hauv cov metabolism ntawm folic acid, uas yog qhov tseem ceeb rau kev sib txuas DNA thiab kev faib tawm ntawm tes. Qhov kev ua no pab txhawm rau txhawm rau tiv thaiv kab mob thiab txo qhov mob.
2. Cov lus qhia:
Apremilast: Feem ntau siv rau kev kho mob ntawm psoriatic mob caj dab thiab cov quav hniav psoriasis.
Methotrexate: Nrog nws txoj kev siv ntau yam, methotrexate tau muab tshuaj los kho qee yam mob, xws li mob caj dab rheumatoid, psoriasis, thiab lwm yam kab mob.

3. Kev saib xyuas:
Apremilast: Kev saib xyuas tsis tu ncua rau cov kev mob tshwm sim yog qhov tseem ceeb, thiab nws yuav tsis tas yuav tsum tau kuaj xyuas ntau zaus piv rau methotrexate.
Methotrexate: suav nrog kev cuam tshuam tsis zoo ntawm daim siab thiab pob txha pob txha, yuav tsum tau saib xyuas ntau zaus ntawm daim siab ua haujlwm thiab suav ntshav.
Dab tsi yog Tshuaj Apremilast siv rau
Apremilast hmoovyog ib qho tshuaj siv los kho qee yam kab mob inflammatory, tshwj xeeb tshaj yog cov kab mob autoimmune. Nws raug cais raws li phosphodiesterase 4 (PDE4) inhibitor. Feem ntau siv hauv:
1. Psoriatic mob caj dab
Cov kab mob sib kis mob ntev hu ua psoriatic mob caj dab feem ntau coexist nrog psoriasis. Cov tawv nqaij mob tsis tu ncua hu ua psoriasis yog typified los ntawm thaj ua rau thaj liab ntawm daim tawv nqaij saum npoo npog hauv cov nplai dawb-dawb. Psoriatic mob caj dab yog tus cwj pwm los ntawm qhov tsis xis nyob thiab o nyob rau hauv cov pob qij txha me me ntawm cov ntiv tes thiab cov ntiv taw thiab qhov chaw liab liab thiab sov sov nyob ib ncig ntawm thaj chaw cuam tshuam. Nws kuj tuaj yeem ua rau cov pob qij txha tawv thaum sawv ntxov lossis tom qab ncua sij hawm tsis ua haujlwm thiab cov ntsia hlau txawv txav, xws li pitting, grooving, lossis thickening. Cov yam ntxwv ntawm caj ces, ib puag ncig, thiab kev tiv thaiv kab mob hauv lub cev tuaj yeem cuam tshuam rau kev tsim tus kab mob. Inhibiting PDE-4 txo cov kev tsim cov tshuaj kho mob, tshwj xeeb tshaj yog nyob rau hauv cov qe ntshav dawb. Tsis tas li ntawd, nws muaj peev xwm tswj tau cov synthesis ntawm inflammatory mediators xws li interleukin -17 (IL-17), interferon- (IFN- ), thiab qog necrosis factor- (TNF- ). Cov yam ntxwv no muaj feem xyuam rau cov kab mob ntawm cov kab mob psoriatic mob caj dab, yog li nws cov teebmeem tuaj yeem pab txo qhov mob thiab pob qij txha o thiab txhim kho cov tsos mob ntawm tus neeg mob.
Nov yog qee qhov kev tshawb fawb txog nws hauv kev kho mob psoriatic mob caj dab:
PALACE Trial: Cov kev sim no suav nrog PALACE 1, PALACE 2, thiab PALACE 3. Cov txiaj ntsig tau pom tias nws muaj txiaj ntsig zoo dua li cov placebo hauv kev txhim kho cov tsos mob ntawm tus mob caj dab thiab cov neeg mob ua haujlwm thiab txo cov tsos mob ntawm daim tawv nqaij psoriasis.
Kev sim ESTEEM: Kev Ua Tau Zoo thiab Kev Nyab Xeeb Kev Ntsuas Kev Ntsuas Cov Teebmeem ntawm nws hauv psoriasis. Qhov kev foob feem ntau tsom rau nws cov txiaj ntsig ntawm kev kho psoriasis. Thaum qhov kev sim ESTEEM feem ntau tsom rau kev ntsuas qhov cuam tshuam ntawm nws ntawm cov kab mob psoriatic tawv nqaij, qhov kev sim kuj suav nrog qee qhov kev ntsuam xyuas ntawm psoriatic mob caj dab vim psoriatic mob caj dab sib koom nrog cov kab mob ntawm daim tawv nqaij. Nws tau pom cov txiaj ntsig zoo hauv kev txhim kho ob qho tib si ntawm daim tawv nqaij thiab cov tsos mob ntawm kev mob caj dab.

2. Plaque psoriasis
Plaque psoriasis lesions feem ntau yog liab, me ntsis tsa cov plaques them nrog silvery-dawb nplai. Cov plaques tuaj yeem tshwm sim nyob txhua qhov ntawm lub cev tab sis feem ntau nyob ib ncig ntawm lub luj tshib, hauv caug, tawv taub hau, sab nraub qaum, thiab pelvis. Plaque psoriasis tuaj yeem ua rau muaj kev hloov pauv hauv qhov tsos thiab khaus, tsis xis nyob, lossis kub hnyiab. Kev tiv thaiv kab mob ua haujlwm tsis zoo ua rau cov kab mob inflammatory, mob tawv nqaij mob psoriasis. Ntau yam xws li noob caj noob ces, kev tiv thaiv kab mob tsis zoo, ib puag ncig, thiab kev ua neej yuav cuam tshuam rau nws qhov pib. Los ntawm kev tiv thaiv PDE-4 enzyme los ntawm kev ua haujlwm, nws yuav txo qis kev tsim cov kab mob inflammatory (xws li leukocyte interleukin -17, interferon- , thiab qog necrosis factor- ), uas tuaj yeem txo qhov mob thiab txo cov tsos mob ntawm qhov chaw ntawm qhov txhab.
Nyob rau hauv lub pathogenesis ntawm psoriasis, txawv txav ua kom lub cev tiv thaiv kab mob ua rau kom ceev ceev kev loj hlob thiab shedding ntawm daim tawv nqaij hlwb, tsim plaque zoo li daim tawv nqaij lesions. Alpresin tuaj yeem cuam tshuam ntawm qib cellular los ntawm kev tswj hwm thiab txo qis kev tsim cov inflammatory mediators: kab mob kev loj hlob thiab kev loj hlob. Tsis tas li ntawd, nws txoj kev kho mob muaj peev xwm rau psoriasis tuaj yeem cuam tshuam nws txoj kev cuam tshuam ntawm lub cev tiv thaiv kab mob thiab kev tsiv teb tsaws.
Nov yog qee qhov kev sim nrog nws hauv cov quav hniav psoriasis:
Kev sim LIBERATE: Txoj kev tshawb no ntsuas qhov kev kho mob zoo rau cov tib neeg uas muaj cov quav hniav me me psoriasis. Cov txiaj ntsig tau qhia tias nws txo qhov mob ntawm daim tawv nqaij thiab cov tsos mob tsawg dua piv rau cov placebo.
Kev sim PSOR-005: Qhov kev sim no yog txhawm rau ntsuas kev nyab xeeb thiab kev ua tau zoo ntawm cov tshuaj hauv cov neeg uas muaj plaque psoriasis hnyav. Cov txiaj ntsig tau sim ua pov thawj cov txiaj ntsig ntawm nws hauv kev txhim kho daim tawv nqaij qhov txhab thiab txo qis kev tsis xis nyob.

Hoobkas
1. Xi'an Sonwu Biotech Co., Ltd muaj lub Hoobkas tsim, tsim khoom, thiab khaws cov khoom, yog li nws muaj cov khoom tsim nyog. Xi'an Sonwu muaj kev txiav txim kom zoo, huv si, thiab huv si ntau lawm. Nyob rau hauv Xi'an Sonwu, cov kws tshawb fawb tuaj yeem tsim cov khoom tshiab zoo.
2. Xi'an Sonwu muaj cov cai nruj rau cov neeg ua haujlwm faib los ntawm kev tsim khoom thiab kev sim rau kev muag khoom. Txhawm rau kom ntseeg tau tias txhua yam khoom raug thauj mus los, kev txhawb nqa cov ntaub ntawv nruj thiab kev pabcuam tom qab muag tau muab.

Daim ntawv pov thawj

Pob

Logistics

Dhau li lav cov khoom, lwm qhov tseem ceeb tshaj plaws yog cov neeg siv khoom tuaj yeem tau txais cov khoom zoo. Yog li, Xi'an Sonwu muab txhua yam kev xa khoom raws li kev xav tau sib txawv.

FAQ
Cov koob tshuaj pom zoo ntawm nws hauv psoriasis thiab psoriatic mob caj dab yog:
psoriatic mob caj dab
Pib koob tshuaj: 30 milligrams (mg) ob zaug ib hnub.
Cov koob tshuaj kho mob: Txhawm rau kom tau txais kev saib xyuas zaum kawg, nce ntxiv ntawm qhov pib koob tshuaj mus rau 30 mg ob zaug ib hnub.
plaque psoriasis
Pib koob tshuaj: 30 mg ob zaug ib hnub.
Cov koob tshuaj kho mob: Txhawm rau kom tau txais kev saib xyuas zaum kawg, nce ntxiv ntawm qhov pib koob tshuaj mus rau 30 mg ob zaug ib hnub.
Yog tias koj xav paub 99 hmoov apremilast lwm tus neeg, koj tuaj yeem tiv tauj Xi'an Sonwu. Nyem rau email, thiab tom qab ntawd koj tau txais cov khoom zooapremilast hmoov.
Email:sales@sonwu.com
Cim npe nrov: apremilast hmoov, Tuam Tshoj, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, nqe, tej, ntshiab, raw, mov, kev muag khoom














