Telmisartan yog dab tsi
Telmisartan hmoovyog ib tug ntev-acting antagonist ntawm angiotensin II hom 1 (AT II) receptors uas yog siv los kho mob ntshav siab. Nws muaj antihypertensive, tiv thaiv ntshav qab zib, tiv thaiv rog, tiv thaiv kab mob, thiab tiv thaiv hyperlipidemic kev ua ub no. Thiab nws txo qis cov roj (cholesterol) tag nrho thiab LDL hauv vivo thiab nws kuj txo qhov hnyav nce thiab nce kev ua haujlwm siab thiab siv oxygen hauv lwm yam tsiaj qauv. Qhov sib xyaw no kuj yog ib qho kev xaiv ntawm PPAR / δ, txo qis insulin, piam thaj, thiab triglyceride qib hauv cov rog rog noj cov nas. Hauv cov hlwb endothelial, Nws txo qis kev qhia ntawm MCP-1 thiab VCAM-1 thiab tiv thaiv kev ua kom NF-κB.

Nws yog cov tshuaj uas muaj nyob rau hauv chav kawm ntawm angiotensin II receptor antagonists. Nws yog feem ntau siv rau kev kho mob ntshav siab thiab tseem tuaj yeem muab tshuaj los tiv thaiv cov xwm txheej hauv plawv hauv cov neeg mob uas muaj qee yam kev pheej hmoo. Nws ua haujlwm los ntawm kev thaiv cov kev ua ntawm angiotensin II uas yog ib yam tshuaj uas ua rau cov hlab ntsha nqaim, yog li txo cov ntshav siab.
Nws muaj nyob rau hauv daim ntawv ntawm cov hmoov, uas yuav yaj nyob rau hauv dej los yog lwm yam kua rau kev tswj tau yooj yim. Qhov ntau npaum thiab lub sijhawm yuav txawv nyob ntawm tus neeg mob thiab cov lus teb rau cov tshuaj. Nws yog ib qho tseem ceeb uas yuav tsum tau ua raws li cov tshuaj noj thiab sab laj nrog tus kws kho mob.
COA
|
Kev tsom xam |
Specification |
Kev tshwm sim |
|
Aρpearance |
Dawb hmoov |
Ua raws |
|
tsw |
Yam ntxwv |
Ua raws |
|
Assay |
Ntau dua lossis sib npaug li 99 feem pua |
99.71% ua |
|
Melting point |
261 ~ 263 degree |
261.3 degree |
|
Poob rau ziab |
Tsawg dua lossis sib npaug li 5.0 feem pua |
2.38 feem pua |
|
Tshauv |
Tsawg dua lossis sib npaug li 5.0 feem pua |
2.65 feem pua |
|
Hnyav Hlau |
Tsawg dua lossis sib npaug li 10ppm |
Ua raws |
|
Raws li |
Tsawg dua lossis sib npaug li 1ppm |
Ua raws |
|
Pb |
Tsawg dua lossis sib npaug li 2ppm |
Ua raws |
|
Hg |
Tsawg dua lossis sib npaug rau 0.1ppm |
Ua raws |
|
Cd |
Tsawg dua lossis sib npaug li 1ppm |
Ua raws |
|
Microbiological |
||
|
Tag Nrho Phaj suav |
Tsawg dua lossis sib npaug li 1000cfu / g |
Ua raws |
|
Poov & Pwm |
Tsawg dua lossis sib npaug li 100cfu / g |
Ua raws |
|
Salmonella |
Tsis zoo |
Tsis zoo |
|
E. Coli |
Tsis zoo |
Tsis zoo |
|
Tshuaj tua kab residue |
Tsis zoo |
Tsis zoo |
|
Xaus |
Ua raws li Enterprise Standard |
|
Qhov twg yuav Telmisartan
Xi'an Sonwu Biotech Co. Ltd. muaj kev paub dhau los hauv kev lag luam thoob ntiaj teb thiab kev noj qab haus huv kev lag luam. Insisting rau txoj kev ntseeg raws li kev ntseeg thiab zoo ua ntej yog peb lub tuam txhab txoj cai. Peb nruj me ntsis tswj cov khoom zoo, uas txhais tau tias kev xaiv pib los ntawm raw cov ntaub ntawv. Tsis tas li ntawd, peb tuav txhua qhov kev nthuav dav thiab txo cov nqi mus rau qhov siab tshaj plaws, thiab tom qab ntawd peb cov neeg siv khoom tuaj yeem tau txais cov khoom lag luam zoo. Raws li cov no, cov neeg siv khoom tau muab cov lus pom zoo rau peb cov khoom. Yog li koj tuaj yeem nrhiav Xi'an Sonwu Biotech Co. Ltd. thaum koj xav yuav Telmisartan.
Xi'an Sonwu ua kom paub tseeb ntawm cov khoom zoo, yog li cov qauv tuaj yeem muab tau. Ntawm no yog qhov ntau.
|
Daim ntawv |
Tus Qauv Zauv |
Yam tsawg kawg nkaus |
|
Hmoov |
50g |
100g |
Dab tsi yog Qhov Teeb Meem
Nws yog ib hom tshuaj uas siv los kho cov ntshav siab (hypertension) thiab qee yam mob plawv. Zoo li txhua yam tshuaj,Telmisartan hmoovtej zaum yuav muaj kev phiv tshwm sim. Nov yog qee qhov kev mob tshwm sim uas tau tshaj tawm:
1. kiv taub hau: Nws tuaj yeem ua rau kiv taub hau lossis tsis pom kev, tshwj xeeb tshaj yog thaum koj sawv ntawm qhov chaw zaum lossis pw. Nws yog ib qho tseem ceeb uas yuav tsum tau maj mam nce kom txo tau qhov kev pheej hmoo ntawm kev ntog.
2. Kev qaug zog: Qee tus neeg yuav muaj kev nkees lossis qaug zog thaum noj nws. Yog tias cov tsos mob tshwm sim los yog mob hnyav, nws raug nquahu kom sab laj nrog kws kho mob.

3. Mob taub hau: Mob taub hau yog ib qho kev mob tshwm sim ntawm Telmisartan. Txawm li cas los xij, yog tias mob taub hau hnyav los yog tsis tu ncua, nws raug nquahu kom nrhiav kev kho mob.
4. Teeb meem plab: Tej zaum nws yuav ua rau muaj teeb meem hauv plab hnyuv xws li xeev siab, raws plab, lossis mob plab. Yog tias cov tsos mob no ua teeb meem, kev sab laj nrog tus kws kho mob pom zoo.

5. Hypotension: Nws tuaj yeem ua rau cov ntshav siab poob qis, tshwj xeeb tshaj yog thaum pib kho lossis siv ntau dua. Qhov no tuaj yeem ua rau cov tsos mob xws li kiv taub hau, kiv taub hau, lossis tsis xis nyob. Kev saib xyuas ntshav siab tsis tu ncua yog qhov tseem ceeb.
6. Kev tsis haum tshuaj: Muaj tsawg zaus, cov tib neeg yuav muaj kev fab tshuaj. Cov tsos mob ntawm kev tsis haum tshuaj muaj xws li pob khaus, khaus, o, kiv taub hau hnyav, lossis ua tsis taus pa. Yog tias ib qho ntawm lawv tshwm sim, yuav tsum tau nrhiav kev kho mob tam sim.
Nws yog ib qho tsim nyog sau cia tias cov npe saum toj no tsis yog tag nrho, thiab ib tus neeg cov lus teb rau cov tshuaj tuaj yeem sib txawv. Nws yog ib qho tseem ceeb uas yuav tau sab laj nrog tus kws kho mob rau cov ntaub ntawv tus kheej hais txog cov kev mob tshwm sim raws li koj cov keeb kwm kho mob tshwj xeeb.
Dab tsi tshuaj yuav tsum tsis txhob noj nrog Telmisartan
Zoo li lwm yam tshuaj, nws yuav cuam tshuam nrog qee yam tshuaj, uas tuaj yeem cuam tshuam rau lawv cov txiaj ntsig lossis ua rau muaj kev phiv. Nov yog qee cov piv txwv ntawm cov tshuaj uas yuav tsum tau siv nrog ceev faj lossis zam thaum noj nws:
1. Cov tshuaj uas tsis yog-Steroidal Anti-Inflammatory Drugs (NSAIDs): NSAIDs xws li ibuprofen, naproxen, thiab aspirin tuaj yeem txo cov ntshav siab. Lawv kuj tuaj yeem ua rau muaj teeb meem rau lub raum thaum noj ua ke. Yog tias koj xav tau noj NSAIDs rau qhov mob nyem lossis mob, nws raug nquahu kom sab laj nrog koj tus kws kho mob rau kev taw qhia.
2. Potassium-Sparing Diuretics thiab Potassium Supplements: Kev sib xyaw nrog cov tshuaj potassium-sparing diuretics (xws li, spironolactone, amiloride) lossis cov tshuaj potassium ntxiv tuaj yeem ua rau cov ntshav nce ntxiv, ua rau hyperkalemia. Kev soj ntsuam ze ntawm cov poov tshuaj yog qhov tseem ceeb hauv cov xwm txheej zoo li no.
3. Lithium: Nws tuaj yeem nce qib lithium hauv lub cev, uas ua rau muaj kev phom sij. Yog tias koj noj lithium, koj tus kws kho mob yuav tsum saib xyuas koj cov qib lithium kom ze.
4. Digoxin: Nws tuaj yeem nce qib ntawm digoxin me ntsis (siv los kho mob plawv) hauv cov ntshav. Kev saib xyuas cov qib digoxin tsis tu ncua raug qhia thaum siv tib lub sijhawm.
5. Tej yam tshuaj Antidiabetic: Nws tuaj yeem txhim kho cov ntshav qab zib kom txo qis cov tshuaj xws li insulin lossis tshuaj tiv thaiv kab mob hauv qhov ncauj. Cov neeg mob ntshav qab zib yuav tsum saib xyuas lawv cov ntshav qab zib kom zoo thaum pib lossis hloov kho.
6. Lwm cov tshuaj tiv thaiv ntshav siab: Kev siv ntau yam tshuaj txo cov ntshav siab, suav nrog lwm cov tshuaj angiotensin receptor blockers (ARBs), ACE inhibitors, lossis beta-blockers, tuaj yeem ua rau cov ntshav siab ntau dhau. Kev soj ntsuam kaw thiab hloov koob tshuaj yuav tsim nyog thaum sib xyaw cov tshuaj no.
Qhov no tsis yog ib daim ntawv teev tag nrho, thiab tej zaum yuav muaj lwm yam tshuaj sib cuam tshuam tshwj xeeb rau ib tus neeg mob. Nws yog ib qho tseem ceeb kom qhia rau koj tus kws kho mob txog txhua yam tshuaj, tshuaj, lossis tshuaj ntsuab uas koj noj ua ntej pib cov hmoov no lossis lwm yam tshuaj tshiab.
Yog Telmisartan Thiab Losartan Tib yam
Thaum lawv muaj cov txheej txheem zoo sib xws ntawm kev ua thiab siv rau cov hom phiaj zoo sib xws, muaj qee qhov sib txawv ntawm ob:
1. Kev ua tau zoo: Ob leeg tuaj yeem kho cov ntshav siab thiab txo cov kev pheej hmoo ntawm cov hlab plawv zoo. Txawm li cas los xij, cov lus teb ntawm tus kheej rau cov tshuaj no yuav txawv, thiab ib qho yuav ua tau zoo dua li lwm tus rau ib tus neeg.
2. Lub Sijhawm Ua Haujlwm: Cov hmoov no muaj lub sijhawm ntev ntawm kev ua piv rau losartan. Qhov no txhais tau hais tias nws tuaj yeem muab kev tswj ntshav siab rau lub sijhawm ntev dua tom qab txhaj tshuaj ib zaug, tso cai rau noj ib hnub ib zaug. Losartan feem ntau yuav tsum tau noj ob zaug ib hnub.

3. Muaj Peev Xwm: Nws raug suav hais tias muaj zog tshaj losartan raws li nws lub peev xwm los thaiv cov angiotensin II receptors, ua rau kom ntshav siab ntau dua.
4. Metabolism: Losartan yog metabolized los ntawm lub siab mus rau hauv ib qho active metabolite hu ua E3174, uas ua rau nws cov teebmeem. Telmisartan, ntawm qhov tod tes, feem ntau metabolized los ntawm lub siab yam tsis tsim cov metabolites tseem ceeb.
5. Cov Lus Qhia Pom Zoo: Cov hmoov no tau pom zoo rau kev kho mob ntshav siab thiab txo cov kev pheej hmoo ntawm cov hlab plawv, nrog rau lub plawv nres thiab mob stroke. Losartan yog siv los kho cov ntshav siab thiab txo cov kev pheej hmoo ntawm mob stroke, tshwj xeeb tshaj yog cov neeg uas muaj ntshav siab thiab sab laug ventricular hypertrophy.
Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias kev xaiv ntawm lawv yuav tsum tau ua raws li tus neeg mob yam xwm txheej, xws li keeb kwm kev kho mob, kev zam, thiab kev teb rau kev kho mob. Tus kws kho mob tuaj yeem txiav txim siab cov tshuaj tsim nyog tshaj plaws rau ib tus neeg tshwj xeeb.
Lisinopril vs Telmisartan
Ob leeg yog cov tshuaj siv los kho cov ntshav siab (hypertension) thiab qee yam mob plawv. Lawv koom nrog cov chav kawm sib txawv ntawm cov tshuaj antihypertensive thiab muaj qee qhov sib txawv:
1. Mechanism of Action: Lisinopril yog ib qho angiotensin-hloov enzyme (ACE) inhibitor, uas ua haujlwm los ntawm inhibiting enzyme. Cov enzyme no hloov angiotensin I mus rau angiotensin II. Telmisartan, ntawm qhov tod tes, yog angiotensin II receptor blocker (ARB), uas thaiv qhov kev txiav txim ntawm angiotensin II ntawm nws cov receptors.

2. Muaj peev xwm: Nws feem ntau suav hais tias muaj zog ntau dua los thaiv cov teebmeem ntawm angiotensin II piv rau lisinopril. Txawm li cas los xij, cov lus teb ntawm tus kheej yuav txawv, thiab qhov ua tau zoo ntawm txhua yam tshuaj tuaj yeem nyob ntawm qhov xwm txheej xws li tus neeg mob tus mob thiab lawv cov lus teb rau kev kho mob.
3. Lub Sijhawm Ua Haujlwm: Nws muaj lub sijhawm ua haujlwm ntev dua piv rau lisinopril. Qhov no txhais tau hais tias cov hmoov no muab kev tswj ntshav siab rau lub sijhawm ntev dua tom qab txhaj tshuaj ib zaug, tso cai rau noj ib hnub ib zaug. Lisinopril feem ntau yuav tsum tau noj ib hnub ib zaug lossis ob zaug-hnub noj hauv qee kis.
4. Cov teebmeem tshwm sim: Ob leeg ntawm lawv yuav ua rau muaj kev phiv, txawm hais tias cov kev mob tshwm sim tshwj xeeb tuaj yeem sib txawv ntawm tib neeg. Cov kev mob tshwm sim ntawm lisinopril tuaj yeem muaj xws li hnoos, kiv taub hau, mob taub hau, thiab cov tsos mob plab. Cov hmoov no yuav ua rau muaj kev phiv xws li kiv taub hau, qaug zog, mob taub hau, thiab mob plab. Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias cov kev mob tshwm sim loj heev tsis tshua muaj tab sis ua tau nrog ob qho tshuaj.
5.Combination Therapy: Ob leeg tuaj yeem siv ua ke nrog lwm cov tshuaj tiv thaiv kab mob siab kom tswj ntshav siab zoo dua thaum tsim nyog. Txawm li cas los xij, kev sib xyaw ua ke ntawm ACE inhibitor zoo li lisinopril nrog ARB zoo li telmisartan feem ntau tsis pom zoo rau kev pheej hmoo ntawm kev phiv.
Kev xaiv ntawm lawv yuav tsum tau ua raws li tus neeg mob yam tseem ceeb, suav nrog keeb kwm kev kho mob, cov yam ntxwv tshwj xeeb kub siab, thiab cov lus teb rau kev kho mob. Tus kws kho mob tuaj yeem ntsuas tus neeg mob thiab muab cov lus qhia tshwj xeeb txog cov tshuaj uas tsim nyog tshaj plaws.
Vim li cas Telmisartan Noj Hmo Hmo
Kev noj hmo thaum hmo ntuj yog ib qho kev pom zoo, txawm hais tias nws yuav txawv nyob ntawm tus kheej thiab cov lus qhia ntawm tus kws kho mob. Qhov laj thawj tom qab noj nws thaum hmo ntuj yog feem ntau cuam tshuam nrog nws cov tshuaj pharmacokinetics, cov qauv ntshav siab, thiab ua kom cov tshuaj muaj txiaj ntsig zoo. Nov yog qee qhov laj thawj:
1. Kev tswj ntshav siab: Cov ntshav siab siab tshaj plaws thaum sawv ntxov thaum sawv ntxov, yog li kev pheej hmoo ntawm plawv nres lossis mob stroke thaum lub sijhawm no nce ntxiv. Telmisartan, thaum noj hmo, tuaj yeem muab 24- teev tswj ntshav siab, pab tswj cov ntshav siab kom ruaj khov nyob rau ib hnub, suav nrog cov sijhawm sawv ntxov tseem ceeb.
2. Circadian Rhythm: Cov hmoov no muaj txiaj ntsig zoo tuaj yeem cuam tshuam los ntawm lub cev circadian atherosclerosis, uas tswj ntau yam txheej txheem physiological dhau ntawm 24- teev voj voog. Kev noj tshuaj thaum hmo ntuj ua raws li kev hloov pauv hauv cov ntshav siab thiab tuaj yeem txhim kho nws qhov cuam tshuam rau renin-angiotensin system, uas koom nrog hauv kev tswj ntshav siab.

3. Dosing Convenience: Nws muaj lub sijhawm ntev ntawm kev txiav txim, tso cai rau noj ib hnub ib zaug. Noj thaum hmo ntuj tuaj yeem yooj yim dua rau ntau tus neeg, vim tias lawv tuaj yeem muab tso rau hauv lawv cov kev ua hmo ntuj lossis ua ntej yuav mus pw.
4. Cov Lus Teb Rau Tus Kheej: Qee tus neeg yuav muaj ntshav siab ntau dua thaum noj thaum hmo ntuj piv rau lwm lub sijhawm nruab hnub. Cov lus teb no tuaj yeem sib txawv ntawm cov tib neeg, thiab nws yog qhov tseem ceeb uas yuav tsum ua raws li cov lus qhia ntawm tus kws kho mob hais txog lub sijhawm zoo ntawm kev tswj hwm tshuaj.
Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias kev txiav txim siab noj telmisartan thaum hmo ntuj yuav tsum tau tham nrog tus kws kho mob. Lawv tuaj yeem txiav txim siab txog tus kheej, xws li tus neeg mob cov qauv ntshav siab, kev tswj hwm tshuaj, thiab kev noj qab haus huv tag nrho, txhawm rau txiav txim siab txog kev noj tshuaj kom tsim nyog.
Hoobkas
1. Xi'an Sonwu Biotech Co., Ltd muaj nws lub Hoobkas, yog li nws muaj cov khoom tsim nyog. Tsis tas li, Xi'an Sonwu muaj chav ua haujlwm huv thiab huv si nrog cov cuab yeej siv siab heev. Nrog cov thawj coj ntawm Xi'an Sonwu, cov kws tshawb fawb tau tsim cov khoom tshiab los ua kom tau raws li cov neeg siv khoom xav tau.
2. Xi'an Sonwu Biotech Co., Ltd muaj cov cuab yeej ntsuas qib siab thiab cov kws tshaj lij, uas txhua tus qhia tias Xi'an Sonwu lub hom phiaj muab cov ntaub ntawv raug thiab ua tau zoo thiab cov kev pabcuam zoo.


Daim ntawv pov thawj

Pob

Logistics Hloov tshiab

Ntxiv nrog rau kev lees paub cov khoom zoo, lwm qhov tseem ceeb tshaj plaws yog cov neeg tuaj yeem tau txais cov khoom lag luam zoo. Yog li, Xi'an Sonwu muab txhua yam kev xa khoom raws li kev xav tau sib txawv.

Vim Li Cas Xaiv Peb
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Peb lub tuam txhab muaj 10- xyoo dhau los hauv kev tsim khoom, tsim khoom, thiab muag khoom.
Peb lub tuam txhab muaj cov kws tshaj lij nrog kev faib cov neeg ua haujlwm kom meej.
Peb muaj cov kws tshaj lij thiab cov cuab yeej siv los xyuas kom meej cov khoom zoo.
Cov khoom raug kuaj los ntawm cov neeg thib peb.
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