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Tetracaine Hydrochloride hmoov

Tetracaine Hydrochloride hmoov

Cov tsos mob: Dawb crystalline hmoov
Specification: 99%
CAS: 136-47-0
Cov roj formula: C15H25ClN2O2
Molecular Luj: 300.824
Txee Lub neej: 2 Xyoo Kev Cia Siab
Tshuag: Tsim nyog Tshuag
Daim ntawv pov thawj: COA, ISO, GMP, HACCP, SGS
Kev Pabcuam: Kev Pabcuam OEM (Pub Private Package)

Khoom Taw qhia

 

Tetracaine HCl
Tetracaine hydrochloride hmoovyog siv los loog qhov chaw ntawm lub cev thaum lub sij hawm kho mob thiab phais cov txheej txheem, thiab nws yog ib qho tshuaj loog hauv zos. Nws zoo txo ​​qhov mob hauv qhov chaw tsom los ntawm kev tiv thaiv cov paj hlwb los ntawm kev nkag mus rau hauv lub cev. Nws yog feem ntau siv hauv kev kho mob xws li ophthalmology, kho hniav, thiab dermatology los pab txo qhov tsis xis nyob thiab mob hauv cov neeg mob uas tau phais. Nws yog ib tus tswv cuab ntawm ester tshuaj loog tsev neeg ntawm cov tshuaj loog hauv zos thiab tau siv dav vim nws qhov pib ua haujlwm sai thiab lub sijhawm luv ntawm kev ua. Nws cov kev siv tseem ceeb yog subarachnoid, epidural, paj hlwb, thiab mucosal nto tshuaj loog. Piv txwv li, hauv kev phais hniav, tetracaine Hcl tuaj yeem siv rau hauv qhov ncauj mucosa rau kev siv tshuaj loog hauv zos ntawm lub qhov ntswg thiab caj pas thiab tseem siv ua ntej ntau yam kev kuaj mob endoscopic los tiv thaiv laryngeal thiab esophageal reflux. Nyob rau hauv ophthalmology, nws yog siv rau intraocular siab ntsuas, corneal microscopy, tshem tawm thiab suturing ntawm corneal txawv teb chaws lub cev, ntau yam kev ntsuam xyuas thiab kuaj mob ntawm ophthalmology, thiab tshuaj loog hauv zos rau me me kev phais. Nws lub peev xwm los tsim tshuaj loog sai sai ua rau nws muaj txiaj ntsig thaum xav tau kev kho mob sai. Yog tias koj txaus siab rau cov khoom siv tshuaj loog, xws li lidocaine, procaine, thiab lwm yam, thov hu rau Xi'an Sonwu. Xi'an Sonwu tuaj yeem muab tetracaine HCL hmoov rau koj.

Tetracaine HCl structure

 

Certificate Of Analysis

Cov khoom

Specification

Cov txiaj ntsig

Qhov tshwm sim

Dawb crystalline hmoov

Ua raws

Kev txheeb xyuas

ABC in pass

Ua raws

Solubility

Soluble hauv dej

Dissolve hauv ethanol

DMSO: Ntau dua lossis sib npaug rau 30mg / mL (99.73 mM)

Ua raws

USP Reference cov qauv

USP Tetracaine Hydrochloride RS, USP Endotoxin RS.

Ua raws

Melting point

149 degree

149 degree

Chromatographic purity

Hauv Pass

Ua raws

Muaj feem xyuam

Tsis ntau tshaj qhov kev daws teeb meem 0.05%

Ua raws

Cov hlau hnyav

Tsawg dua lossis sib npaug li 10ppm

Ua raws

PH

Residue ntawm ignition

4.5-6.5

5.8

Tsawg dua lossis sib npaug rau 0.10%

0.05%

Poob rau ziab

Tsawg dua los yog sib npaug rau 0.5%

0.19%

Assay

98.0 -101.0%

100.1%

 

Qhov twg Yuav Tetracaine HCl
Xi'an Sonwu Biotech Co. Ltd. muaj ntau tshaj kaum xyoo ntawm kev lag luam kev lag luam, tshwj xeeb hauv kev tsim thiab muag cov ntaub ntawv raw. Xi'an Sonwu tau tsim kev sib koom tes ruaj khov thiab txhim khu kev qha nrog cov teb chaws hauv Asmeskas, Asia, Europe, thiab Oceania. Xi'an Sonwu muab cov khoom zoo ua ntej thiab siv zog los muab txhua tus neeg siv khoom nrog cov kev pabcuam zoo kom tau raws li lawv cov kev xav tau tag nrho.
Txhua theem ntawm Xi'an Sonwu cov txheej txheem tsim khoom, pib nrog kev xaiv cov khoom siv raw, nruj nruj tswj hwm. Cov khoom lag luam zoo yog Xi'an Sonwu qhov tseem ceeb tshaj plaws, thiab lub tuam txhab kev mob siab rau kev ua tiav tau pom nyob rau hauv txhua yam ntawm nws cov haujlwm, suav nrog kev xaiv cov khoom siv raw, cov txheej txheem tsim khoom, cov qauv kuaj, thiab cov neeg ua haujlwm tshaj lij. Xi'an Sonwu tuaj yeem txo cov nuj nqis yam tsis muaj kev txi zoo los ntawm kev ua tib zoo saib xyuas txhua yam, lav tias cov neeg tau txais cov khoom muaj txiaj ntsig zoo kawg li.
Xi'an Sonwu zoo siab rau cov lus pom zoo uas nws tau txais los ntawm cov neeg siv khoom, uas tau lees paub qhov zoo ntawm cov khoom. Txhawm rau ua pov thawj ntxiv cov khoom lag luam, Xi'an Sonwu yuav muab cov qauv rau koj los kuaj.

Daim ntawv

Tus Qauv Zauv

Yam tsawg kawg nkaus

Hmoov

100g

100g


Cov neeg siv khoom 'Cov lus pom zoo

-801

 

Tetracaine Hydrochloride siv rau dab tsi
1. Ophthalmology
Tetracaine hydrochloride nquag siv hauv ophthalmology los tshuaj loog lub qhov muag (cornea) nto rau kev kuaj thiab cov txheej txheem xws li kev ntsuas intraocular siab, tshem tawm lub cev txawv teb chaws, lossis kev cuam tshuam me me. Nws zoo meej rau cov kev siv no vim tias nws pib ua haujlwm sai thiab sijhawm txaus. Nws yuav raug siv los muab tshuaj loog hauv zos kom txo tau cov neeg mob tsis xis nyob thaum lub sij hawm kuaj mob los yog lub teeb nyem los yog thaum kuaj ntshav siab. Ophthalmologists siv nws los txo tus neeg mob qhov mob thaum tshem tawm cov khoom txawv teb chaws ntawm lub qhov muag saum npoo los yog pob txha. Tej zaum nws yuav raug txiav txim siab thaum kho lossis tshuaj xyuas lub pob txha raug mob los ntawm kev puas tsuaj, nrog rau thaum lub sij hawm kho qhov muag pom kev phais xws li LASIK (laser hauv situ keratomileusis) lossis PRK (nto txheej laser keratomileusis).

 

2. Kev kho hniav
Tetracaine Hcl tuaj yeem siv los ua tshuaj loog rau ntawm lub qhov ncauj mucosa los muab lub sijhawm luv luv rau kev kho cov pos hniav, kho kab mob, lossis lwm yam txheej txheem uas yuav ua rau mob. Qhov ntawd yog qhov tshwj xeeb tshaj yog thaum kho qhov chaw rhiab lossis ua cov txheej txheem uas yuav ua rau tsis xis nyob rau tus neeg mob. Nws kuj tseem tuaj yeem siv los ua ib txoj kev kho mob ib ntus los pab tswj kev mob hnyav los ntawm cov teeb meem hniav (xws li cov hniav tawg, cov pos hniav, thiab lwm yam) thaum tos kev kho hniav ntxiv.

Dentistry

 

3. Otolaryngology
Tetracaine Hcl tuaj yeem siv rau cov txheej txheem qhov ntswg xws li qhov ntswg qhov ntswg, tshem tawm qhov ntswg, thiab kho epistaxis. Kev siv cov tshuaj pleev ib ce tuaj yeem txo tus neeg mob qhov mob thiab tsis xis nyob thaum ua haujlwm no. Thaum ua laryngoscopy, kev phais lub suab, lossis lwm yam kev kho mob laryngeal, Tetracaine Hcl tuaj yeem siv los ua tshuaj loog los pab txo qhov mob hauv lub ntsws, txo cov hnoos qeev thiab tsis xis nyob, thiab ua rau kev phais lossis kev kuaj mob zoo dua. Txawm hais tias nws muaj tsawg dua kev siv otological ncaj qha, nws yuav siv tau los txo qhov mob thaum lub sij hawm phais me me los yog cov txheej txheem kuaj mob, xws li kev ntxuav pob ntseg los yog tshem tawm lub cev txawv teb chaws.

 

Dab tsi yog Hom Kev Ua Ntawm Tetracaine
Tetracaine hydrochloride hmoovyog ib qho tshuaj loog hauv zos uas ua haujlwm los ntawm kev thaiv kev sib kis ntawm cov paj hlwb. Nws tshwm sim los ntawm inhibiting influx ntawm sodium ions los ntawm ion channels nyob rau hauv lub paj hlwb membrane. Los ntawm kev ua tiav qhov kev thaiv no, tetracaine zoo thaiv kev tsim khoom thiab kev ua haujlwm ntawm cov hlab ntsha impulses. Thaum kawg, qhov no ua rau muaj qhov tsis xis nyob hauv cheeb tsam thiab qhov mob nyem cuam tshuam nrog kev noj nws.
Tetracaine belongs rau tsev neeg tshuaj loog hauv zos ester thiab nquag siv hauv ntau cov txheej txheem kho mob kom txo tau qhov mob thiab tsis xis nyob. Nws ua rau cov hlab ntsha xaus thiab qhov hnov ​​​​tsw receptors hauv thaj chaw tsom thaum siv. Nws ua haujlwm los ntawm kev khi rau ib qho tshwj xeeb sodium ion channel uas pom nyob rau hauv daim nyias nyias ntawm cov paj hlwb. Blocks sodium channels uas yog voltage-gated thiab tam sim no nyob rau hauv neuronal daim nyias nyias. Tetracaine stabilizes neuronal daim nyias nyias thiab txwv tsis pub muaj peev xwm los ntawm kev pib thiab kis los ntawm kev txuas mus rau tej qhov chaw ntawm cov channel. Qhov kev thaiv no inhibits kev ua ntawm cov hlab ntsha impulses, zoo loog ntawm thaj chaw uas tetracaine tau tswj hwm. Tetracaine tshwj xeeb tiv thaiv cov kab hluav taws xob-gated sodium los ntawm kev qhib, uas yog qhov tseem ceeb rau kev pib thiab nthuav tawm cov peev txheej hauv cov paj hlwb. Nres lub peev xwm ntawm daim nyias nyias los ntawm kev nce mus rau qhov pib xav tau los tsim kom muaj peev xwm ua tau, thaiv lub hlwb lub peev xwm kom tau txais cov cim mob. Qhov ntawd tshwm sim vim hais tias sodium channel blockade tiv thaiv qhov kev txiav txim muaj peev xwm lub depolarization theem, uas yog ib qho tseem ceeb rau kev nthuav tawm ntawm cov hlab ntsha impulses raws li lub paj hlwb. Raws li qhov tshwm sim, cov paj hlwb hauv thaj chaw thov tsis tuaj yeem xa cov cim kev hnov ​​​​lus, ua rau muaj tshuaj loog ib ntus thiab mob nyem. Tsis tas li ntawd, nws cov teebmeem yog thim rov qab. Thaum cov tshuaj metabolized los yog diffused deb ntawm cov paj hlwb, cov sodium channel rov ua haujlwm li qub, cia cov paj hlwb mus ncig thiab hnov ​​​​qab mus rau thaj chaw.
Tsis tas li ntawd, tetracaine hom kev txiav txim siab yog nyob ntawm concentration. Cov concentrations siab dua thaiv impulses los ntawm kev hnov ​​​​lus thiab lub cev muaj zog neurons, ua rau tsis hnov ​​​​tsw ( tshuaj loog ) thiab cov leeg tuag tes tuag taw hauv thaj tsam ntawm daim ntawv thov. Tsawg concentrations feem ntau cuam tshuam rau kev hnov ​​​​mob neurons, ua rau muaj kev ua xua yam tsis muaj lub cev muaj zog.

mode of action of tetracaine hcl

Factors cuam tshuam nws cov nyhuv:
pH thiab cov ntaub so ntswg ib puag ncig: Qhov pib thiab lub sijhawm ntawm kev ua haujlwm tuaj yeem cuam tshuam los ntawm pH ntawm cov ntaub so ntswg thiab muaj lwm yam tshuaj, xws li vasoconstrictors, uas qee zaum koom ua ke los ua kom cov nyhuv ntawm tetracaine los ntawm kev txo nws txoj kev nqus.

Lipid Solubility: Tetracaine yog lipid-soluble ntau dua li qee cov tshuaj loog hauv zos, tso cai rau nws nkag mus rau cov paj hlwb zoo dua, pab txhawb rau nws cov tshuaj loog muaj zog.

Protein Binding: Nws txoj kev sib raug zoo rau plasma proteins thiab cov ntaub so ntswg tuaj yeem cuam tshuam rau nws cov tshuaj pharmacokinetics, suav nrog nws qhov pib, lub sijhawm ua haujlwm, thiab cov metabolism.

 

Puas yog Tetracaine thiab Lidocaine Tib yam
Tetracaine thiab lidocaine yog ob qho tib si tshuaj loog hauv zos. Tetracaine yog ib qho ester ntawm cov tshuaj loog hauv zos thiab feem ntau siv tau zoo thiab kav ntev dua lidocaine. Qhov ntawd ua rau tetracaine haum rau kev phais uas yuav tsum tau siv tshuaj loog ntev. Nws yog feem ntau siv rau tshuaj loog ntawm qhov muag (ophthalmology), qhov ntswg, caj pas, thiab txha caj qaum. Nws muaj zog dua thiab ua haujlwm ntev dua tso cai rau nws siv rau hauv cov txheej txheem tshwj xeeb, tab sis nws kuj muaj kev pheej hmoo siab dua ntawm cov kab mob toxicity yog tias siv carelessly. Lidocaine yog ib feem ntawm cov tshuaj loog hauv zos amide chav kawm. Nws tsis tshua muaj zog thiab muaj lub sijhawm luv luv ntawm kev ua haujlwm tshaj li tetracaine, tab sis nws tseem siv tau rau ntau daim ntawv thov. Lidocaine feem ntau muaj cov tshuaj toxicity tsawg dua li tetracaine, ua rau nws haum rau ntau yam kev siv. Lidocaine tau siv dav hauv ntau qhov chaw kho mob, suav nrog cov txheej txheem kho hniav, kev phais me, thiab cov khoom siv tshuaj pleev ib ce.
Lawv lub ntsiab sib txawv yog nyob rau hauv chemical class; tetracaine yog ester, thaum lidocaine yog amide. Qhov sib txawv no cuam tshuam rau lawv cov metabolism thiab, qee qhov, kev pheej hmoo ntawm kev tsis haum tshuaj. Amides (xws li lidocaine) feem ntau tsis tshua muaj kev ua xua ntau dua li esters (xws li tetracaine). Lidocaine feem ntau metabolized hauv daim siab, thaum plasma esterases hydrolyze tetracaine thiab metabolized hauv daim siab. Vim nws lub zog ntau dua, tetracaine feem ntau raug xaiv rau cov txheej txheem uas yuav tsum tau ua kom tob tob lossis ua kom ntev ntev. Nyob rau tib lub sijhawm, lidocaine muaj qhov pib ua haujlwm sai dua thiab tsis muaj zog, ua rau nws tsim nyog rau ntau yam ntawm cov txheej txheem luv luv. Tsis tas li ntawd, thaum muab piv nrog procaine, lwm yam tshuaj loog, tetracaine hydrochloride, muaj roj ntau dua solubility dua procaine, kev nkag mus ntau dua li procaine, thiab cov tshuaj loog hauv zos yog kaum npaug ntau dua procaine.

Lidocaine

 

Hoobkas
1. Xi'an Sonwu Biotech Co., Ltd muaj nws lub Hoobkas los tsim, tsim, thiab khaws cov khoom, yog li muaj cov khoom tsim nyog. Xi'an Sonwu muaj kev txiav txim kom zoo, huv si, thiab huv si ntau lawm. Nyob rau hauv Xi'an Sonwu, cov kws tshawb fawb tuaj yeem tsim cov khoom tshiab zoo.
2. Xi'an Sonwu muaj cov cai nruj rau cov neeg ua haujlwm faib los ntawm kev tsim khoom thiab kev sim rau kev muag khoom. Tag nrho cov khoom escorting yog lav los ntawm nruj cov ntaub ntawv txhawb nqa thiab kev pab cuam tom qab muag.

302

 

Daim ntawv pov thawj

303


Pob

304


Logistics

-802
Dhau li lav cov khoom, lwm qhov tseem ceeb tshaj plaws yog cov neeg siv khoom tuaj yeem tau txais cov khoom zoo. Yog li, Xi'an Sonwu muab txhua yam kev xa khoom raws li kev xav tau sib txawv.

FAQ
Cov tshuaj twg yog tetracaine hydrochloride feem ntau siv nrog?
epidural thaiv
Qhov xav tau concentration yog {{0}}.15%-0.3% tov, ua ke nrog lidocaine hydrochloride; qhov siab tshaj plaws yog 0.3%, qhov ntau npaum li cas ntawm ib zaug yog 40-50mg, thiab qhov siab tshaj plaws yog 80mg.
subarachnoid thaiv
Feem ntau siv sib tov (1% tetracaine hydrochloride 1ml tov nrog 10% qabzib 1ml thiab 13% ephedrine hydrochloride 1ml), cov koob tshuaj ib txwm siv rau ib zaug yog 10mg, 15mg yog qhov txwv, thiab 20mg yog qhov siab tshaj plaws.
Yog tias koj xav paub cov chaw tsim khoom tetracaine Hcl, koj tuaj yeem tiv tauj Xi'an Sonwu. Nyem rau email, thiab tom qab ntawd koj tau txais cov khoom zootetracaine hydrochloride hmoov.
Email:sales@sonwu.com

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