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Lubiprostone hmoov

Lubiprostone hmoov

Cov tsos mob: Dawb Crystal hmoov
Specification: NLT 98%
CAS: 333963-40-9
Cov roj formula: C20H32F2O5
Molecular Luj: 390.462 g / mol
Txee Lub neej: 2 Xyoo Kev Cia Siab
Tshuag: Tsim nyog Tshuag
Daim ntawv pov thawj: ISO, GMP, HACCP SGS
Kev Pabcuam: OEM Kev Pabcuam (Piv txwv pob, Capsules)

Khoom Taw qhia

 

Lubiprostone yog dab tsi

Lubiprostone hmoovyog ib hom tshuaj siv los kho mob cem quav thiab chim siab plob tsis so tswj nrog cem quav (IBS-C) rau cov neeg laus. Nws yog ib hom kab mob plab uas ua rau kom cov kua dej tso rau hauv cov hnyuv, ua rau cov quav mos thiab ua kom yooj yim dua.

 

Lubiprostone yog cais raws li cov tshuaj chloride channel activator thiab ua rau cov tshuaj chloride hauv cov hnyuv epithelium hlwb, uas pab ua kom cov kua dej tso rau hauv cov hnyuv lumen. Qhov no ua rau kom muaj zog ntawm cov hnyuv, ua rau kev txhim kho plab hnyuv.

 

Nws muaj txiaj ntsig zoo hauv kev txo cov tsos mob ntawm cem quav ntev thiab IBS-C hauv kev sim tshuaj. Cov teebmeem thib ob muaj xws li xeev siab, raws plab, mob plab, thiab flatulence. Tsawg dua tab sis cov kev mob tshwm sim hnyav dua tuaj yeem ua rau muaj kev tsis haum tshuaj, plab hnyuv perforation, thiab electrolyte imbalances.

 

Nws yuav tsum tsis txhob siv rau cov poj niam cev xeeb tub lossis pub niam mis, vim tias nws txoj kev nyab xeeb hauv cov neeg no tsis tau tsim. Nws kuj yuav tsum tau siv nrog ceev faj rau cov neeg mob uas muaj keeb kwm ntawm plab hnyuv, kab mob plab, lossis kab mob raum lossis kab mob siab.

 

Hauv cov ntsiab lus, lubiprostone yog cov tshuaj siv los kho mob cem quav thiab IBS-C hauv cov neeg laus los ntawm kev ua kom cov kua dej tso rau hauv cov hnyuv. Nws muaj nyob rau hauv daim ntawv capsule rau kev tswj qhov ncauj thiab feem ntau yog noj ob zaug ib hnub nrog zaub mov thiab dej. Thaum feem ntau ua tau zoo, nws tuaj yeem ua rau muaj kev phiv thiab yuav tsum tau siv ceev faj hauv cov neeg mob tshwj xeeb.

 

 

Lubiprostone powder mf

 

Certificate of Analysis

SAIB

SPECIFICATION

TSEEM CEEB

Qhov tshwm sim

Dawb los yog dawb dawb hmoov hmoov

Ua raws

Kev txheeb xyuas

Los ntawm IR

Ua raws

Los ntawm HPLC

Ua raws

Solubility

Soluble nyob rau hauv DMF, sparingly soluble nyob rau hauv THF, me ntsis soluble nyob rau hauv methanol thiab acetonitrile, heev sightly soluble nyob rau hauv ethanol thiab dichloromethane, insoluble nyob rau hauv dej

Ua raws

Polymorphic Form

Polymorphic daim ntawv 1

Ua raws

Melting Point

211ºC~216ºC

212.8ºC~214.9ºC

Cov ntsiab lus dej

Tsawg dua lossis sib npaug rau 0.50%

0.10%

Hnyav Hlau

Tsawg dua lossis sib npaug li 20ppm

Ua raws

Residue ntawm Ignition

Tsawg dua lossis sib npaug rau 0.20%

0.09%

Yam khoom

Ib qho impurity: Tsawg dua lossis sib npaug rau 0.10%

0.06%

Tag nrho cov impurities: Tsawg dua lossis sib npaug rau 1.00%

0.16%

Assay

(ntawm lub hauv paus anhydrous)

98.0%~102.0%

99.94%

Particle Loj

D90: Tsawg dua lossis sib npaug rau 100µm

Ua raws

 

Yuav Qhov twg

Xi'an Sonwu Biotech Co., Ltd. muaj kev paub nplua nuj hauv kev lag luam thoob ntiaj teb thiab kev lag luam kev noj qab haus huv. Hais txog kev ntseeg raws li kev ntseeg thiab ua ntej yog peb lub tuam txhab txoj cai. Peb nruj me ntsis tswj cov khoom zoo, uas txhais tau tias kev xaiv pib los ntawm raw khoom. Tsis tas li ntawd, peb tuav txhua qhov kev nthuav dav thiab txo tus nqi mus rau qhov siab tshaj plaws, ces peb cov neeg siv khoom tuaj yeem tau txais cov khoom lag luam zoo. Raws li cov no, cov neeg siv khoom tau muab cov lus pom zoo rau peb cov khoom. Yog li nrhiav Xi'an Sonwu Biotech Co. Ltd. thaum koj xav tau cov khoom no.

 

Peb ua kom paub tseeb tias cov khoom zoo, yog li cov qauv tuaj yeem muab tau. Ntawm no yog qhov ntau.

Daim ntawv

Tus Qauv Zauv

Yam tsawg kawg nkaus

Hmoov

10g

10g

 

Cov neeg siv khoom zoo lus

comment

 

Kev Pabcuam OEM

Xi'an Sonwu tsis tsuas yog tuaj yeem muab cov khoom zoolubiprostone hmoov, tab sis kuj muab lwm yam ntaub ntawv.

Yog li txhua tus neeg siv khoom tuaj yeem hloov kho yam lawv xav tau. Thiab cov khoom hauv qab no tuaj yeem muab tau.

Customized capsules shells (loj, xim, khoom)

Customized fwj (loj, xim, khoom, style)

Customized ntim (nqus foil ntim, thawv, nruas)

Customized daim ntawv lo (xim zaj duab xis, matte zaj duab xis, daim npog qhov muag)

 

Dab tsi yog Mechanism Ntawm Kev Ua Ntawm Lubiprostone

Lubiprostone yog tus neeg saib xyuas mob plab uas siv los kho mob idiopathic cem quav thiab chim siab plob tsis so tswj nrog cem quav (IBS-C) rau cov neeg laus. Nws ua haujlwm los ntawm kev ua kom cov kua dej tso rau hauv cov hnyuv, ua rau cov quav softer thiab yooj yim dua. Cov tshuaj muaj nyob rau hauv chav kawm ntawm cov tshuaj hu ua chloride channel activators, uas tseem hu ua pro-secretory agents.

 

Cov txheej txheem ntawm kev txiav txim ntawm lubiprostone cuam tshuam nrog kev ua kom cov chloride channel uas muaj nyob rau hauv lub apical membrane ntawm txoj hnyuv epithelium. Cov kab no yog lub luag haujlwm rau kev zais cov tshuaj chloride ions rau hauv lumen ntawm txoj hnyuv. Cov chloride ions tsim ib qho osmotic gradient, ua rau dej txav mus rau hauv lub lumen thiab ua kom muaj kua dej ntau ntxiv.

 

Lubiprostone xaiv khi thiab qhib hom -2 chloride channels (ClC-2) nyob rau ntawm qhov chaw apical ntawm txoj hnyuv epithelial hlwb. Kev ua kom cov kab no ua rau cov chloride ions tso rau hauv lub lumen ntawm txoj hnyuv, uas, dhau los, txhawb kev tso dej thiab electrolytes rau hauv lumen. Qhov txiaj ntsig no yog ua kom cov quav mos thiab ua kom nws cov khoom ntau, ua kom yooj yim dua.

 

Ntxiv rau nws cov teebmeem ntawm cov tshuaj chloride, lubiprostone tau pom tias muaj lwm yam kev ua haujlwm uas yuav ua rau nws cov teebmeem kev kho mob. Piv txwv li, nws tau raug tshaj tawm tias inhibit qhov kev ua ntawm sodium-hydrogen exchanger -3 (NHE3) transporter, uas yog lub luag haujlwm rau kev nqus ntawm sodium thiab dej hauv txoj hnyuv. Los ntawm inhibiting NHE3, lubiprostone tuaj yeem txhim kho qhov tso tawm ntawm dej thiab electrolytes rau hauv lub lumen.

 

Lubiprostone kuj tau pom tias txhawb kev tsim cov prostaglandins, ib txwm muaj cov tshuaj uas tswj hwm ntau yam txheej txheem physiological, suav nrog kev mob plab hnyuv. Prostaglandins paub tias yuav ua kom muaj cov tshuaj chloride thiab dej tso rau hauv cov hnyuv lumen, uas tuaj yeem ua rau muaj kev cuam tshuam rau lubiprostone.

 

Nyob rau hauv cov ntsiab lus, lubiprostone yog ib tug kab mob plab hnyuv siab raum uas xaiv activates chloride raws nyob rau hauv lub apical nto ntawm txoj hnyuv epithelial hlwb. Qhov no ua rau lub zais ntawm chloride ions mus rau hauv lub lumen ntawm txoj hnyuv, uas nyob rau hauv lem txhawb lub secretion ntawm dej thiab electrolytes mus rau hauv lub lumen, uas ua rau kom cov kua secretion thiab softer quav. Lubiprostone kuj tseem muaj lwm cov txheej txheem ntawm kev ua, suav nrog inhibition ntawm NHE3 thiab kev txhawb nqa ntawm prostaglandin ntau lawm, uas tuaj yeem txhim kho nws cov teebmeem kev zais cia ntxiv.

 

Lubiprostone powder mechanism

 

Lubiprostone yog Prostaglandin

Lubiprostone tsis yog prostaglandin. Nws yog ib tug hluavtaws derivative ntawm ib txwm tshwm sim bicyclic fatty acid uas ua raws li ib tug xaiv chloride channel activator nyob rau hauv lub plab zom mov. Prostaglandins, ntawm qhov tod tes, yog ib pawg ntawm lipid compounds uas tau los ntawm fatty acids thiab muaj ntau yam cuam tshuam rau lub cev, suav nrog kev tswj kev mob, ntshav khiav, thiab tsim cov ntshav txhaws.

 

Thaum lubiprostone txhawb kev tsim cov prostaglandins hauv plab hnyuv mucosa, nws tsis yog nyob rau hauv cov chav kawm prostaglandin ntawm cov tebchaw. Hloov chaw, nws siv nws cov tshuaj pharmacological ncaj qha los ntawm kev ua kom cov chloride tshwj xeeb hauv cov apical membrane ntawm lub plab hnyuv epithelium.

 

Ua kom cov chloride channels ua rau muaj cov tshuaj chloride ions mus rau hauv txoj hnyuv lumen, tom qab ntawd los ntawm kev txav dej mus rau hauv lub lumen vim yog osmotic gradient tsim los ntawm cov chloride ions. Qhov no ua rau kom cov kua hauv plab tso tawm, ua rau cov quav mos thiab txhim kho plab hnyuv.

 

Tsis tas li ntawd, lubiprostone tau pom tias muaj qhov nqus dej tsawg, uas txhais tau hais tias nws cov teebmeem feem ntau yog nyob rau hauv lub plab zom mov. Nyob rau hauv sib piv, prostaglandins raug tsim thiab tso tawm thoob plaws hauv lub cev, exerting ntau yam physiological teebmeem.

 

Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias thaum lubiprostone txhawb kev tsim cov prostaglandins hauv plab hnyuv mucosa, nws cov txheej txheem ntawm kev ua feem ntau cuam tshuam nrog kev ua kom ncaj qha ntawm cov tshuaj chloride es tsis ua haujlwm raws li prostaglandin nws tus kheej. Qhov kev sib txawv no yog qhov tseem ceeb hauv kev nkag siab txog cov tshuaj pharmacological tshwj xeeb ntawm lubiprostone thiab nws txawv li cas ntawm prostaglandins.

 

Lubiprostone Cov Kev Pab Cuam Tshuam

Lubiprostone, zoo li ntau cov tshuaj, tuaj yeem muaj cov kev mob tshwm sim. Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias tsis yog txhua tus neeg yuav ntsib cov kev mob tshwm sim no, thiab qee tus neeg yuav muaj cov lus teb sib txawv rau cov tshuaj. Cov kev mob tshwm sim ntawm lubiprostone tej zaum yuav muaj xws li:

 

1. Nausea: Nausea yog ib qho ntawm lubiprostone feem ntau tshaj tawm cov kev mob tshwm sim. Qee cov tib neeg tej zaum yuav mob me me mus rau nruab nrab xeev siab, tshwj xeeb tshaj yog thaum pib cov tshuaj, txawm tias cov tsos mob no feem ntau ploj zuj zus mus.

2. Mob plab: Thaum lubiprostone feem ntau yog siv los kho cem quav, paradoxically, qee zaum nws tuaj yeem ua rau raws plab raws li kev phiv. Qhov no feem ntau pom nyob rau hauv cov neeg uas muaj mob plab plob tsis so tswj nrog cem quav (IBS-C).

3. Mob plab: Qee tus neeg yuav muaj mob plab plab, mob plab, lossis mob thaum noj lubiprostone. Cov tsos mob no feem ntau yog me me mus rau nruab nrab ntawm qhov hnyav.

4. Mob taub hau: Mob taub hau yog lwm qhov kev mob tshwm sim ntawm lubiprostone. Cov tib neeg uas muaj mob hnyav lossis mob taub hau yuav tsum sab laj nrog lawv tus kws kho mob.

5. Flatulence: nce roj lossis flatulence tuaj yeem tshwm sim raws li kev mob tshwm sim ntawm kev kho lubiprostone.

6. ntuav: Qee zaum, ntuav tau qhia tias yog ib qho kev mob tshwm sim ntawm lubiprostone.

 

Hoobkas ib puag ncig

Xi'an Sonwu ntau lawm Hoobkas yog zoo-tsim, huv si, thiab huv si, nrog txaus Tshuag. Raws li kev coj noj coj ua ntawm lub tuam txhab, cov kws tshawb fawb tau hais kom tsim cov khoom tshiab. Cov hauv qab no yog qhov chaw sim ntawm peb lub chaw soj nstuam, cov cuab yeej ntsuas qib siab, thiab cov kws tshaj lij kev sim, nrog tus cwj pwm nruj los muab cov ntaub ntawv tseem ceeb rau peb cov khoom thiab muab peb cov neeg siv khoom nrog kev paub zoo.

 

factory

 

Daim ntawv pov thawj

certificates

 

Ntim

packaging

 

Cov ntaub ntawv logistics

logistics

 

Ntxiv nrog rau kev lees paub cov khoom zoo, lwm qhov tseem ceeb tshaj plaws yog cov neeg tuaj yeem tau txais cov khoom lag luam zoo. Yog li, Xi'an Sonwu muab txhua yam kev xa khoom raws li kev xav tau sib txawv.

 

courier

 

Tuam txhab Profile

Xi'an Sonwu Biotech Co., Ltd. Itd yog cov chaw tsim khoom hauv Suav teb thiab cov khoom lag luam. Nws tau tsim nyob rau hauv 2012, thiab nyob rau hauv Hi-Tech industrial Zone Xi'an nroog, Shannxi xeev, Suav teb. Nws them tag nrho cov xim ntawm txoj kev loj hlob, kev tshawb fawb thiab kev tsim khoom noj khoom haus additives, cog extract, APl thiab lwm yam khoom xyaw ntawm cov khoom kho mob. Peb lub tuam txhab muab tsib yam khoom raw khoom: Anti-hair poob Powders, Nootropic, API, Muscle Building products, Cog Extract. Peb ua siab dawb ntseeg tias qhov chaw ntawm kev koom tes zoo yog cov kev pabcuam zoo tshaj plaws thiab zoo. Yog li, txais tos koj qhov kev nug.

 

Yog xav yuavLubiprostone hmoov, thov hu rau Xi'an Sonwu.

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Cim npe nrov: Lubiprostone hmoov, Tuam Tshoj, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, nqe, tej, ntshiab, raw, mov, kev muag khoom

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